SCHEMBL7415044

SCHEMBL7415044

O=C=C1C(CO)NC(=O)N1OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
MAPT P10636 1/20 0.35
TSHR P16473 1/20 0.34
GDA Q9Y2T3 1/20 0.34
KDM4C Q9H3R0 1/20 0.33
GLA P06280 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HBB P68871 1/20 0.32
ALOX15 P16050 1/20 0.32
HTR2C P28335 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20516433 0.73 GAA (0.49) ALDH1A1MEN1KMT2AKDM4CALOX15
SCHEMBL20516432 0.73 GAA (0.49) ALDH1A1MEN1KMT2AKDM4CALOX15
SCHEMBL16577067 0.68 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2MEN1KMT2AMAPT
SCHEMBL7543136 0.68 MEN1 (0.36) ALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL5871291 0.67 NPC1 (0.39) ALDH1A1SMN1; SMN2
SCHEMBL27733749 0.67 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2HTR2C
SCHEMBL9485689 0.65 FABP7 (0.42) ALDH1A1SMN1; SMN2HTR2C
SCHEMBL20516384 0.65 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AMAPTTSHR
SCHEMBL20516387 0.65 ALDH1A1 (0.51) ALDH1A1MEN1KMT2AMAPTTSHR
SCHEMBL20516416 0.64 CES2 (0.44) MEN1KMT2ATSHRKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6391901-B1 Thrombin inhibitors ELI LILLY AND COMPANY 2002-05-21 US disclosed
EP-1027051-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2001-03-07 EP disclosed
EP-1027051-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-08-16 EP disclosed
WO-1998048804-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed