SCHEMBL7416124

SCHEMBL7416124

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)CCc1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.49
CASP7 P55210 1/20 0.49
CTSL P07711 3/20 0.46
CTSB P07858 3/20 0.46
CTSS P25774 3/20 0.46
CTSD P07339 2/20 0.45
REN P00797 2/20 0.45
CA2 P00918 1/20 0.45
ELANE P08246 1/20 0.43
CASP1 P29466 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9579040 0.93 CASP3 (0.46) CASP3CASP7CTSLCTSBCTSS
SCHEMBL7411626 0.85 CASP1 (0.47) CASP3CASP7RENCA2ELANE
SCHEMBL8492203 0.84 CTSD (0.54) CASP3CASP7CTSLCTSBCTSS
SCHEMBL8366143 0.83 CTSD (0.45) CASP3CASP7CTSD
SCHEMBL8364492 0.82 CTSD (0.48) CASP3CASP7CTSDRENELANE
SCHEMBL7415829 0.81 CTSB (0.56) CASP3CTSLCTSBCTSSREN
SCHEMBL7420909 0.81 CTSB (0.56) CASP3CTSLCTSBCTSSREN
SCHEMBL7420907 0.81 CTSB (0.56) CASP3CTSLCTSBCTSSREN
SCHEMBL7414133 0.81 CTSB (0.56) CASP3CTSLCTSBCTSSREN
SCHEMBL7410781 0.81 CASP1 (0.52) CASP3CASP7CTSLCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed