SCHEMBL741659

SCHEMBL741659

COCCCn1c(C2CCCN(C(=O)OC(C)(C)C)C2)nc2cccc(C(=O)OC)c21

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.42
USP30 Q70CQ3 2/20 0.39
HPGDS O60760 1/20 0.39
P2RX7 Q99572 1/20 0.39
BRD4 O60885 1/20 0.39
ACKR3 P25106 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TRPV3 Q8NET8 1/20 0.38
LMNA P02545 3/20 0.38
TP53 P04637 2/20 0.38
ALOX5AP P20292 1/20 0.38
FEN1 P39748 1/20 0.38
MAPT P10636 2/20 0.38
THRB P10828 1/20 0.38
HDAC4 P56524 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL762848 0.93 BRD4 (0.41) PARP1USP30HPGDSP2RX7BRD4
SCHEMBL740662 0.88 P2RX7 (0.41) PARP1USP30HPGDSP2RX7ACKR3
SCHEMBL740661 0.88 P2RX7 (0.41) PARP1USP30HPGDSP2RX7ACKR3
SCHEMBL741974 0.85 KCNH2 (0.52) HPGDS
SCHEMBL741975 0.85 KCNH2 (0.52) HPGDS
SCHEMBL740873 0.82 SCN9A (0.45) USP30HPGDSTRPV3TP53MAPT
SCHEMBL741590 0.82 CTSB (0.35) LMNAMAPT
SCHEMBL741591 0.82 CTSB (0.35) LMNAMAPT
SCHEMBL762854 0.80 P2RX7 (0.42) HPGDSP2RX7BRD4JAK2JAK1
SCHEMBL740746 0.79 CHRM1 (0.46) PARP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed