SCHEMBL7416623

SCHEMBL7416623

NC(=O)C1(CC2CCCC2)CC1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.41
HSD11B1 P28845 1/20 0.39
EPHX1 P07099 4/20 0.38
SLC1A3 P43003 3/20 0.34
SLC1A2 P43004 3/20 0.34
SLC1A1 P43005 3/20 0.34
PARP15 Q460N3 2/20 0.33
PARP10 Q53GL7 2/20 0.33
CYP2D6 P10635 1/20 0.32
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31
SPHK1 Q9NYA1 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ARG1 P05089 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5081028 0.91 HSD11B1 (0.44) ALOX5HSD11B1SLC1A3SLC1A2SLC1A1
SCHEMBL7421923 0.80 CYP2C19 (0.40) ALOX5EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL3913863 0.75 ALOX5 (0.33) ALOX5CYP2D6
SCHEMBL11346600 0.72 CYP2C19 (0.52) ALOX5EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL6586703 0.72 CYP2C19 (0.52) ALOX5EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL11292307 0.72 CYP4F2 (0.45) EPHX1SLC1A3SLC1A2SLC1A1HPGD
SCHEMBL3543709 0.71 SLC6A9 (0.40) HSD11B1
SCHEMBL27206940 0.70 CYP2C19 (0.36) ALOX5EPHX1SLC1A3SLC1A2SLC1A1
SCHEMBL1053596 0.67 CYP2C19 (0.45) ARG1
SCHEMBL23558591 0.66 JAK2 (0.32) ALOX5HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0707570-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-04-24 EP disclosed
WO-1995000489-A1 ISOQUINOLINE DERIVATIVES AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-01-05 WO disclosed