SCHEMBL7418362

SCHEMBL7418362

CC(C)CC(C(=O)O)N(CCc1ccc(-c2ccc(C(F)(F)F)cc2)cc1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 2/20 0.51
PSEN2 P49810 2/20 0.51
APH1B Q8WW43 2/20 0.51
NCSTN Q92542 2/20 0.51
APH1A Q96BI3 2/20 0.51
PSENEN Q9NZ42 2/20 0.51
MMP2 P08253 2/20 0.42
MMP3 P08254 2/20 0.42
MAOB P27338 1/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MMP13 P45452 2/20 0.39
MMP1 P03956 1/20 0.39
MMP7 P09237 1/20 0.39
MMP9 P14780 1/20 0.39
FDFT1 P37268 2/20 0.39
ADAMTS4 O75173 1/20 0.39
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7427409 0.86 MMP12 (0.46) MMP13
SCHEMBL7420384 0.86 MMP12 (0.46) MMP13
SCHEMBL7425601 0.86 MCHR1 (0.50) MMP2MMP3
SCHEMBL7424796 0.85 HPGD (0.38) MMP3FFAR1
SCHEMBL7424342 0.83 PSEN1 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7424015 0.81 GPR88 (0.42) MMP2MMP9
SCHEMBL7419478 0.81 MMP2 (0.42) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7417897 0.80 FOLH1 (0.45)
SCHEMBL7378945 0.80 MEN1 (0.48) MMP2MMP3MMP1MMP7MMP9
SCHEMBL1661113 0.79 CYP11B1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed