SCHEMBL7419478

SCHEMBL7419478

CC(C)CC(C(=O)O)N(CCc1ccc(-c2cc(Cl)cc(Cl)c2)cc1)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.42
MMP3 P08254 1/20 0.42
ADAMTS5 Q9UNA0 2/20 0.40
FFAR4 Q5NUL3 2/20 0.40
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
S1PR1 P21453 1/20 0.39
S1PR5 Q9H228 1/20 0.39
GRN P28799 2/20 0.38
SORT1 Q99523 2/20 0.38
AKR1C2 P52895 1/20 0.38
AKR1C1 Q04828 1/20 0.38
APP P05067 1/20 0.36
MCHR1 Q99705 1/20 0.36
CHKA P35790 1/20 0.36
MME P08473 1/20 0.36
ACE P12821 1/20 0.36
F7 P08709 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419020 0.88 GRN (0.38) MMP2MMP3ADAMTS5GRNSORT1
SCHEMBL7422595 0.87 RXRA (0.40) ADAMTS5RXRARXRBGRNSORT1
SCHEMBL7428192 0.85 CARM1 (0.46) PPARGPPARAGRNSORT1ALDH1A1
SCHEMBL7424796 0.85 HPGD (0.38) MMP3ADAMTS5PPARGPPARAS1PR1
SCHEMBL7427409 0.84 MMP12 (0.46) MCHR1
SCHEMBL7420384 0.84 MMP12 (0.46) MCHR1
SCHEMBL7425601 0.84 MCHR1 (0.50) MMP2MMP3S1PR1MCHR1MME
SCHEMBL7424617 0.83 MAOB (0.42) FFAR4RXRARXRB
SCHEMBL7426638 0.82 ALDH1A1 (0.43) PPARGPPARAGRNSORT1MCHR1
SCHEMBL7424958 0.81 APP (0.39) MMP3ADAMTS5PPARAGRNSORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed