SCHEMBL7419245

SCHEMBL7419245

CC(C)(CCNC(=O)c1ccccc1)CC(=O)N(Cc1ccccc1)C1(C#N)CCNC1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.41
TMEM97 Q5BJF2 5/20 0.41
CTSS P25774 4/20 0.38
CTSK P43235 2/20 0.38
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
ESRRG P62508 1/20 0.35
CTSL P07711 2/20 0.35
CTSB P07858 1/20 0.35
ALDH1A1 P00352 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7420985 0.91 ALDH1A1 (0.43) SIGMAR1TMEM97ALDH1A1
SCHEMBL7420196 0.83 CTSS (0.36) CTSSCTSKNPC1CTSLCTSB
SCHEMBL7420191 0.72 SNCA (0.34) CTSSCTSKCTSLCTSB
SCHEMBL7021621 0.72 RXFP1 (0.34) CTSSCTSKCTSLCTSB
SCHEMBL7021496 0.71 CTSS (0.41) CTSSCTSKCTSLCTSB
SCHEMBL7413191 0.70 CTSS (0.37) SIGMAR1TMEM97CTSSRAB9ACTSL
SCHEMBL7420982 0.69 CTSL (0.36) CTSSCTSKCTSLCTSBALDH1A1
SCHEMBL7023323 0.69 CTSS (0.42) CTSSCTSKCTSLCTSB
SCHEMBL7419141 0.69 AGER (0.39) SIGMAR1TMEM97
SCHEMBL6565858 0.69 NR1H4 (0.36) CTSSCTSKNPC1RAB9ACTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218372-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2002-07-03 EP disclosed
WO-2001019816-A1 NOVEL SPIROHETEROCYCLIC COMPOUNDS USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed