SCHEMBL8565729

SCHEMBL8565729

COC(=O)CCc1ccc(N2CCN(c3ccc4c(c3)CCN(C(=O)OC(C)(C)C)CC4)C2=O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.45
ESR2 Q92731 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP2C19 P33261 1/20 0.38
JAK2 O60674 2/20 0.37
JAK3 P52333 2/20 0.37
PTK2 Q05397 2/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
GPR119 Q8TDV5 3/20 0.36
ENPP2 Q13822 1/20 0.36
USP30 Q70CQ3 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8559518 0.86 HRH3 (0.41) SMN1; SMN2CYP2C19HDAC1TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL8564996 0.85 HRH3 (0.40) SMN1; SMN2CYP2C19HDAC1TMEM97SIGMAR1
SCHEMBL8559578 0.82 HTR6 (0.42) HDAC1DRD2
Hydrochloric Acid SCHEMBL8566255 0.81 HTR6 (0.41) MAPTHDAC1DRD2
SCHEMBL8562720 0.80 S1PR1 (0.45) CYP2C19HDAC1TMEM97SIGMAR1DRD2
SCHEMBL8563370 0.79 ASIC3 (0.40) HDAC1
SCHEMBL7389941 0.78 S1PR1 (0.43) LMNAGPR119
SCHEMBL7473247 0.78 NR1H2 (0.47) NR1H2ESR2NPC1RAB9ALMNA
SCHEMBL7419930 0.77 NR1H2 (0.49) NR1H2ESR2NPC1RAB9ALMNA
SCHEMBL7284346 0.77 HDAC1 (0.39) HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed