SCHEMBL7420320

SCHEMBL7420320

CC(C)C(NC(=O)O)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(=O)C(F)(F)C(=O)NCc1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
REN P00797 6/20 0.50
CYP1A2 P05177 1/20 0.48
CYP2D6 P10635 1/20 0.48
MAPT P10636 1/20 0.48
TSHR P16473 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ELANE P08246 1/20 0.46
PGA5 P0DJD9 1/20 0.46
ALDH1A1 P00352 1/20 0.45
MME P08473 1/20 0.44
ACE P12821 1/20 0.44
CPA1 P15085 1/20 0.44
ACE2 Q9BYF1 1/20 0.44
HTRA1 Q92743 5/20 0.44
CA2 P00918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9421813 0.91 MME (0.48) MMEACECPA1ACE2HTRA1
SCHEMBL7414303 0.88 CMA1 (0.52) SMN1; SMN2ELANEMMEACECPA1
SCHEMBL8364492 0.88 CTSD (0.48) RENELANEPGA5
SCHEMBL8736216 0.84 CTSD (0.53) MMEACECPA1ACE2HTRA1
SCHEMBL7420852 0.82 CMA1 (0.52) RENTSHRPGA5ALDH1A1MME
SCHEMBL7418725 0.81 MME (0.46) MMEACECPA1ACE2HTRA1
SCHEMBL7418157 0.81 REN (0.45) RENELANEPGA5MMEACE
SCHEMBL7423864 0.81 REN (0.45) RENELANEPGA5MMEACE
SCHEMBL7416869 0.80 MME (0.43) RENMMEACECPA1ACE2
SCHEMBL8945318 0.80 CTSD (0.46) MMEACECPA1ACE2HTRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773926-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-05-21 EP claimed
WO-1996002499-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-02-01 WO claimed
WO-1996002499-A1 DIFLUOROSTATONE ANTIVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-02-01 WO disclosed