SCHEMBL7422285

SCHEMBL7422285

CC(C)CC(NCC(C(=O)O)c1csc(-c2cc(Cl)cc(Cl)c2)n1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.47
GRN P28799 3/20 0.44
SORT1 Q99523 3/20 0.44
SHMT1 P34896 2/20 0.41
SHMT2 P34897 2/20 0.41
TLR7 Q9NYK1 1/20 0.37
ACE2 Q9BYF1 4/20 0.37
ACE P12821 3/20 0.37
ADRB2 P07550 2/20 0.35
ADRB1 P08588 2/20 0.35
ADRB3 P13945 2/20 0.35
MAPK1 P28482 1/20 0.35
PDE5A O76074 1/20 0.35
LDHA P00338 1/20 0.35
LDHB P07195 1/20 0.35
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 2/20 0.34
HTT P42858 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426736 0.88 CTSK (0.48) CTSKSORT1SHMT1SHMT2MAPK1
SCHEMBL1655302 0.86 CTSK (0.62) CTSKGRNSORT1PDE5ALDHA
SCHEMBL7425252 0.84 CTSK (0.54) CTSKPDE5ALDHALDHBLMNA
SCHEMBL7424365 0.83 GRN (0.43) CTSKGRNSORT1SHMT1SHMT2
SCHEMBL7426448 0.82 GRN (0.44) GRNSORT1ACE2ACEADRB2
SCHEMBL7420772 0.80 ALDH1A1 (0.51) CTSKSHMT1SHMT2TLR7MAPK1
SCHEMBL7423860 0.80 SORT1 (0.44) GRNSORT1ACE2ACEADRB2
SCHEMBL7382345 0.79 CTSK (0.41) CTSKGRNSORT1MAPK1PDE5A
SCHEMBL7417883 0.78 CTSK (0.55) CTSKPDE5ALDHALDHBMAPT
SCHEMBL7424643 0.78 CTSK (0.39) CTSKSHMT1SHMT2ACE2ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed