SCHEMBL7422935

SCHEMBL7422935

CC(C)CC(NCC(C(=O)O)c1csc(-c2ccc3c(c2)CCO3)n1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PLA2G10 O15496 1/20 0.53
NPC1 O15118 2/20 0.52
RAB9A P51151 2/20 0.52
CLK1 P49759 2/20 0.52
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 1/20 0.45
DNM1L O00429 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
CTSK P43235 1/20 0.43
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
CHEK1 O14757 11/20 0.42
KMT2A Q03164 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5870572 0.82 PLA2G10 (0.55) PLA2G10NPC1RAB9ACLK1KDM4E
SCHEMBL5869975 0.82 PLA2G10 (0.55) PLA2G10NPC1RAB9ACLK1KDM4E
SCHEMBL1655302 0.80 CTSK (0.62) NPC1RAB9AKDM4ESMN1; SMN2CTSK
SCHEMBL7425252 0.79 CTSK (0.54) NPC1RAB9AKDM4ESMN1; SMN2CTSK
SCHEMBL7426736 0.78 CTSK (0.48) KDM4EALDH1A1SMN1; SMN2CTSKTAS1R3
SCHEMBL7422285 0.77 CTSK (0.47) KDM4EALDH1A1SMN1; SMN2CTSK
SCHEMBL7420772 0.76 ALDH1A1 (0.51) KDM4EALDH1A1SMN1; SMN2CTSKKMT2A
SCHEMBL7422924 0.73 PLA2G10 (0.53) PLA2G10NPC1RAB9ACLK1KDM4E
SCHEMBL7417883 0.72 CTSK (0.55) NPC1RAB9AKDM4ESMN1; SMN2CTSK
SCHEMBL7382345 0.71 CTSK (0.41) NPC1RAB9AALDH1A1SMN1; SMN2CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed