SCHEMBL7423101

SCHEMBL7423101

CS(=O)(=O)N[C@H](CCC(=O)O)C(=O)NCCCCc1ccc(C=NN)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR2 O95136 1/20 0.38
S1PR1 P21453 1/20 0.38
S1PR3 Q99500 1/20 0.38
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
PTPN1 P18031 2/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ITGB3 P05106 2/20 0.37
ITGA2B P08514 2/20 0.37
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNB4 P30926 1/20 0.36
CHRNA3 P32297 1/20 0.36
CHRNA4 P43681 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995579 0.85 ITGB3 (0.41) S1PR2S1PR1S1PR3LMNATSHR
SCHEMBL7418987 0.83 LMNA (0.41) S1PR2S1PR1S1PR3LMNATSHR
SCHEMBL7423093 0.83 ITGB3 (0.54) ITGB3ITGA2B
SCHEMBL7423099 0.83 ITGB3 (0.54) ITGB3ITGA2B
SCHEMBL8995577 0.82 MMP12 (0.39) LMNATSHRPTPN1CYP2D6CYP2C9
SCHEMBL8995575 0.82 MMP12 (0.39) LMNATSHRPTPN1CYP2D6CYP2C9
SCHEMBL7415259 0.79 FOLH1 (0.52) CA1CA2KMT2A
SCHEMBL8995553 0.79 FOLH1 (0.52) CA1CA2KMT2A
SCHEMBL8995559 0.78 KMT2A (0.44) S1PR2S1PR1LMNATSHRCYP2D6
SCHEMBL7385812 0.77 S1PR1 (0.49) S1PR1LMNATSHRCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5552431-A ANTICOAGULANTS G. D. SEARLE & CO. (US) 1996-09-03 US disclosed
US-5424334-A Peptide mimetic compounds useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1995-06-13 US disclosed
WO-1993012074-A1 PEPTIDE MIMETIC COMPOUNDS USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1993-06-24 WO disclosed