SCHEMBL7423261

SCHEMBL7423261

CC(C)[C@H](NC(=O)CNS(=O)(=O)CCc1ccccn1)C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)CCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.47
CASP1 P29466 1/20 0.45
CA2 P00918 2/20 0.41
KMT2A Q03164 2/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
MMP1 P03956 1/20 0.38
MMP7 P09237 1/20 0.38
MMP8 P22894 1/20 0.38
MMP12 P39900 1/20 0.38
MMP13 P45452 1/20 0.38
REN P00797 1/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CTSD P07339 1/20 0.37
CASP3 P42574 1/20 0.37
CASP7 P55210 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423302 0.84 CASP1 (0.52) ELANECASP1CTSDCASP3HTRA1
SCHEMBL7411626 0.83 CASP1 (0.47) ELANECASP1CA2KMT2ASMN1; SMN2
SCHEMBL9579040 0.80 CASP3 (0.46) ELANECASP1CA2SMN1; SMN2CYP1A2
SCHEMBL7415944 0.80 CASP1 (0.47) ELANECASP1CA2KMT2ASMN1; SMN2
SCHEMBL7416124 0.79 CASP3 (0.49) ELANECASP1CA2RENCTSD
SCHEMBL7415572 0.79 CASP1 (0.54) CASP1CTSDCASP3HTRA1
SCHEMBL7418534 0.78 ELANE (0.49) ELANEKMT2ASMN1; SMN2CYP1A2MMP1
SCHEMBL7414375 0.78 ELANE (0.49) ELANEKMT2ASMN1; SMN2CYP1A2MMP1
SCHEMBL9578947 0.76 CA2 (0.47) CASP1CA2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7410781 0.75 CASP1 (0.52) ELANECASP1CA2RENCTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO claimed
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed