SCHEMBL7415944

SCHEMBL7415944

CNC(=O)N(CC(=O)N[C@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)C(F)(F)CCc1ccccc1)C(C)C)Cc1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.47
CA2 P00918 2/20 0.47
SMN1; SMN2 Q16637 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
CTSD P07339 4/20 0.38
REN P00797 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
ELANE P08246 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7410782 0.89 CASP1 (0.48) CASP1CA2ALDH1A1ELANE
SCHEMBL7413833 0.88 CASP1 (0.47) CASP1CTSDALDH1A1ELANE
SCHEMBL9579040 0.80 CASP3 (0.46) CASP1CA2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7423261 0.80 ELANE (0.47) CASP1CA2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7411626 0.80 CASP1 (0.47) CASP1CA2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL9578947 0.80 CA2 (0.47) CASP1CA2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7416124 0.77 CASP3 (0.49) CASP1CA2CTSDRENELANE
SCHEMBL7415572 0.75 CASP1 (0.54) CASP1CTSD
SCHEMBL7334046 0.75 CA2 (0.48) CASP1CA2SMN1; SMN2CYP1A2CYP2D6
SCHEMBL7423302 0.74 CASP1 (0.52) CASP1CTSDELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO claimed
US-5256677-A Enzyme inhibitor for treating acquired immune deficiency syndrome ABBOTT LABORATORIES (US) 1993-10-26 US disclosed
WO-1992017176-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1992-10-15 WO disclosed
US-5151438-A Enzyme inhibitors for treatment of aids ABBOTT LABORATORIES (US) 1992-09-29 US disclosed