SCHEMBL7423334

SCHEMBL7423334

Cc1cc(C)cc(Cc2csc(C(CNC(CC(C)C)C(=O)O)C(=O)O)n2)c1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP2C19 P33261 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
MEN1 O00255 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
MMP2 P08253 1/20 0.33
MAPK1 P28482 1/20 0.33
SORT1 Q99523 2/20 0.33
MAPT P10636 1/20 0.33
ITGB1 P05556 2/20 0.33
ITGA4 P13612 2/20 0.33
PTPRB P23467 1/20 0.33
CTSK P43235 1/20 0.32
GRN P28799 1/20 0.32
PYGL P06737 1/20 0.32
MME P08473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7417825 0.88 GRN (0.43) DHFRALDH1A1MAPK1SORT1MAPT
SCHEMBL7424812 0.84 SMN1; SMN2 (0.34) ALDH1A1CYP2C19TAS1R3TAS1R1MEN1
SCHEMBL7426920 0.83 CTSK (0.38) DHFRALDH1A1CYP2C19TAS1R3TAS1R1
SCHEMBL7425447 0.79 DHFR (0.34) DHFRALDH1A1CYP2C19TAS1R3TAS1R1
SCHEMBL7420461 0.76 BCHE (0.37) ALDH1A1MEN1KMT2AMMP2MAPK1
SCHEMBL7426736 0.76 CTSK (0.48) ALDH1A1CYP2C19TAS1R3TAS1R1MEN1
SCHEMBL5869842 0.76 ACE2 (0.39) ALDH1A1CYP2C19TAS1R3TAS1R1MEN1
SCHEMBL8430007 0.76 ACE2 (0.39) ALDH1A1CYP2C19TAS1R3TAS1R1MEN1
SCHEMBL7429293 0.76 SORT1 (0.34) DHFRALDH1A1CYP2C19TAS1R3TAS1R1
SCHEMBL7426239 0.76 MEN1 (0.43) ALDH1A1MEN1KMT2ASORT1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed