Phenylguanidine

Phenylguanidine

SCHEMBL7425328

N=C(N)Nc1ccccc1.O=C(O)C(F)(F)F.O=C(O)C(F)(F)F

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHIT1 Q13231 1/20 0.49
F2 P00734 2/20 0.48
TMPRSS6 Q8IU80 1/20 0.48
KLK1 P06870 3/20 0.48
KLK5 Q9Y337 2/20 0.48
MAPT P10636 2/20 0.47
GAA P10253 1/20 0.47
GFER P55789 1/20 0.47
TP53 P04637 2/20 0.47
TSHR P16473 2/20 0.47
EPHX1 P07099 1/20 0.47
EPHX2 P34913 1/20 0.47
CDK9 P50750 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
PDK1 Q15118 2/20 0.46
PDK2 Q15119 2/20 0.46
PDK3 Q15120 2/20 0.46
PDK4 Q16654 2/20 0.46
HDAC3 O15379 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenylguanidine SCHEMBL1950328 0.86 TP53 (0.56) F2KLK1MAPTGAAGFER
Phenylguanidine SCHEMBL300643 0.86 TP53 (0.56) F2KLK1MAPTGAAGFER
Phenylurea SCHEMBL6505098 0.85 MAPT (0.66) CHIT1MAPTGAAGFERTP53
Trifluoroacetic Acid SCHEMBL30725604 0.84 KLK1 (0.51) F2TMPRSS6KLK1KLK5MAPT
Phenylguanidine SCHEMBL8887604 0.84 TP53 (0.54) F2KLK1MAPTGAAGFER
Phenylguanidine SCHEMBL256023 0.84 ALDH1A1 (0.58) F2KLK1MAPTGAAGFER
Phenylguanidine SCHEMBL11154590 0.82 HSD17B10 (0.59) F2KLK1MAPTGAAGFER
Phenylguanidine SCHEMBL28414520 0.82 HSD17B10 (0.52) F2KLK1MAPTGAAGFER
Phenylguanidine SCHEMBL4027020 0.82 ALDH1A1 (0.56) F2KLK1MAPTGAAGFER
Phenylguanidine SCHEMBL29249611 0.82 ALDH1A1 (0.56) F2KLK1MAPTGAAGFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6211228-B1 COMPOUNDS WITH AMINO, GUANIDINO AND AMIDINO HETEROCYCLIC COMPOUNDS AXYS PHARMACEUTICALS, INC 2001-04-03 US disclosed
US-6022969-A Compositions and methods for treating mast-cell mediated conditions AXYS PHARMACEUTICALS, INC. (US) 2000-02-08 US disclosed
EP-0782571-A1 COMPOSITIONS AND METHODS FOR TREATING MAST-CELL INFLAMMATORY CONDITION ARRIS PHARMACEUTICAL CORPORATION (US) 1997-07-09 EP disclosed
WO-1996009297-A1 COMPOSITIONS AND METHODS FOR TREATING MAST-CELL INFLAMMATORY CONDITION ARRIS PHARMACEUTICAL CORPORATION (US) 1996-03-28 WO disclosed