SCHEMBL7425779

SCHEMBL7425779

CC(C)CC(NCC(C(=O)O)c1ccc(-c2cccnc2)cc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 1/20 0.49
CTSK P43235 5/20 0.48
CTSS P25774 5/20 0.48
CTSL P07711 5/20 0.48
AKR1C3 P42330 1/20 0.46
AKR1C2 P52895 1/20 0.46
MKNK1 Q9BUB5 4/20 0.44
MKNK2 Q9HBH9 4/20 0.44
ADRB1 P08588 1/20 0.42
ADRB3 P13945 1/20 0.42
DYRK1A Q13627 1/20 0.41
GPR88 Q9GZN0 1/20 0.40
CTSB P07858 3/20 0.40
DGAT1 O75907 1/20 0.39
SLC2A1 P11166 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424096 1.00 NTSR1 (0.49) NTSR1CTSKCTSSCTSLAKR1C3
SCHEMBL7420389 0.88 CTSS (0.48) CTSKCTSSCTSLAKR1C3AKR1C2
SCHEMBL7427413 0.88 CTSS (0.48) CTSKCTSSCTSLAKR1C3AKR1C2
SCHEMBL7424801 0.83 CTSS (0.46) CTSKCTSSCTSLAKR1C3AKR1C2
SCHEMBL7421360 0.82 GPR132 (0.53)
SCHEMBL7425607 0.82 CTSL (0.48) CTSKCTSSCTSLCTSB
SCHEMBL7378949 0.81 MME (0.50) CTSKCTSS
SCHEMBL7424498 0.81 CTSK (0.49) CTSKCTSSCTSLCTSBDGAT1
SCHEMBL7418370 0.79 PSEN1 (0.60) CTSKCTSSCTSLAKR1C3AKR1C2
SCHEMBL7419482 0.79 GRN (0.49) CTSKCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed