SCHEMBL7426906

SCHEMBL7426906

Cc1cc(C)cc(Cc2nc(CCN(C(=O)O)C(CC(C)C)C(=O)O)cs2)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 3/20 0.37
BCHE P06276 8/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
KLKB1 P03952 1/20 0.30
KLK1 P06870 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423323 0.93 BCHE (0.33) HDAC1HDAC6BCHEMEN1KMT2A
SCHEMBL7424356 0.89 HDAC1 (0.36) HDAC1HDAC6BCHEKMT2A
SCHEMBL7426729 0.83 TP53 (0.39)
SCHEMBL7417819 0.81 HDAC1 (0.34) HDAC1HDAC6BCHEMEN1KMT2A
SCHEMBL7382337 0.81 MAPT (0.41) TDP1
SCHEMBL7429286 0.80 NR4A2 (0.31)
SCHEMBL7425444 0.79 NR4A2 (0.32)
SCHEMBL7424802 0.79 ALDH1A1 (0.36) HDAC1HDAC6
SCHEMBL1655299 0.76 ATM (0.46)
SCHEMBL7418496 0.76 ADRB3 (0.33) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed