SCHEMBL7423323

SCHEMBL7423323

Cc1cc(C)cc(Cc2csc(CCN(C(=O)O)C(CC(C)C)C(=O)O)n2)c1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BCHE P06276 10/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HDAC1 Q13547 7/20 0.31
HDAC6 Q9UBN7 7/20 0.31
TP53 P04637 1/20 0.30
LNPEP Q9UIQ6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426906 0.93 HDAC1 (0.37) BCHEMEN1KMT2ATDP1HDAC1
SCHEMBL7417819 0.88 HDAC1 (0.34) BCHEMEN1KMT2ATDP1HDAC1
SCHEMBL7424802 0.84 ALDH1A1 (0.36) HDAC1HDAC6
SCHEMBL7424356 0.81 HDAC1 (0.36) BCHEKMT2AHDAC1HDAC6
SCHEMBL7425444 0.80 NR4A2 (0.32)
SCHEMBL7426729 0.80 TP53 (0.39) TP53
SCHEMBL7429286 0.79 NR4A2 (0.31)
SCHEMBL7382337 0.77 MAPT (0.41) TDP1
SCHEMBL7420456 0.76 ADRB3 (0.35) MEN1KMT2ALNPEP
SCHEMBL7426234 0.75 LOXL2 (0.47) MEN1KMT2AHDAC1HDAC6TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO claimed
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed