SCHEMBL7426937

SCHEMBL7426937

NC(OC(=O)c1c(Cl)cccc1Cl)C(=O)CCC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC15A1 P46059 1/20 0.42
KMT2A Q03164 2/20 0.38
AKR1B1 P15121 1/20 0.38
FEN1 P39748 1/20 0.37
ALDH1A1 P00352 2/20 0.37
CASP3 P42574 3/20 0.35
KDM4E B2RXH2 1/20 0.35
TXNRD1 Q16881 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
LTA4H P09960 1/20 0.34
MAPT P10636 1/20 0.34
PTK2B Q14289 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
MEN1 O00255 1/20 0.34
RAB9A P51151 1/20 0.34
CASP6 P55212 2/20 0.34
CASP8 Q14790 2/20 0.34
ITGB2 P05107 1/20 0.33
ICAM1 P05362 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8764806 0.72 SLC15A1 (0.44) SLC15A1L3MBTL1RAB9ACASP6NPC1
SCHEMBL8764753 0.71 CASP1 (0.43) KMT2AALDH1A1CASP3MAPTMEN1
SCHEMBL5583677 0.70 FEN1 (0.58) KMT2AAKR1B1FEN1ALDH1A1KDM4E
SCHEMBL12946377 0.70 CASP3 (0.49) KMT2AALDH1A1CASP3TXNRD1TDP1
SCHEMBL11230817 0.69 KMT2A (0.46) KMT2AAKR1B1FEN1ALDH1A1TXNRD1
SCHEMBL9245419 0.69 CA12 (0.66) ALDH1A1SMN1; SMN2MAPTRAB9ANPC1
SCHEMBL21866492 0.69 ALDH1A1 (0.48) KMT2AFEN1ALDH1A1KDM4ETXNRD1
SCHEMBL6801086 0.67 ALDH1A1 (0.63) KMT2AAKR1B1FEN1ALDH1A1CASP3
SCHEMBL18321223 0.66 HCAR2 (0.49) KMT2AALDH1A1SMN1; SMN2MAPTPTK2B
SCHEMBL5703139 0.65 ALDH1A1 (0.58) KMT2AAKR1B1FEN1ALDH1A1TXNRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1091930-A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-04-18 EP disclosed
WO-2000001666-A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2000-01-13 WO disclosed