SCHEMBL8764753

SCHEMBL8764753

C=CCOC(=O)NC(OC(=O)c1c(Cl)cccc1Cl)C(=O)CCC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 16/20 0.43
ALDH1A1 P00352 2/20 0.37
HPGD P15428 1/20 0.37
CASP3 P42574 1/20 0.37
MAPT P10636 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7254765 0.74 CASP3 (0.38) CASP1ALDH1A1HPGDCASP3MEN1
SCHEMBL646188 0.73 CASP1 (0.44) CASP1CASP3
SCHEMBL4439353 0.72 CYP3A4 (0.58) ALDH1A1HPGDMEN1KMT2A
SCHEMBL8764759 0.72 CASP1 (0.47) CASP1CASP3
SCHEMBL7426937 0.71 SLC15A1 (0.42) ALDH1A1HPGDCASP3MAPTMEN1
SCHEMBL645654 0.68 CASP1 (0.48) CASP1CASP3
SCHEMBL1409148 0.68 ALDH1A1 (0.35) CASP1ALDH1A1HPGDCASP3MAPT
SCHEMBL6405747 0.68 CASP1 (0.37) CASP1ALDH1A1HPGDCASP3MEN1
SCHEMBL2217364 0.68 ALDH1A1 (0.35) CASP1ALDH1A1HPGDCASP3MAPT
SCHEMBL13178975 0.68 CASP1 (0.48) CASP1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed