SCHEMBL7427741

SCHEMBL7427741

O=C(O)CC(=O)CC1CCN1C(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
SLC6A9 P48067 1/20 0.41
CNR1 P21554 2/20 0.39
CNR2 P34972 2/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
OPRM1 P35372 6/20 0.39
OPRD1 P41143 6/20 0.39
OPRK1 P41145 6/20 0.39
OPRL1 P41146 6/20 0.39
CACNA2D1 P54289 2/20 0.38
CACNA1B Q00975 2/20 0.38
CACNB1 Q02641 2/20 0.38
CACNA1C Q13936 2/20 0.38
CACNA1H O95180 1/20 0.38
NPC1 O15118 1/20 0.38
CYP2D6 P10635 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9684251 0.89 ALDH1A1 (0.44) ALDH1A1SLC6A9CNR1CNR2OPRM1
SCHEMBL8534618 0.78 OPRM1 (0.46) ALDH1A1OPRM1OPRD1OPRK1OPRL1
Hydrochloric Acid SCHEMBL11268886 0.76 OPRM1 (0.44) ALDH1A1OPRM1OPRD1OPRK1OPRL1
SCHEMBL9682023 0.75 ALDH1A1 (0.47) ALDH1A1OPRM1OPRD1OPRK1OPRL1
SCHEMBL11415783 0.73 MEN1 (0.44) OPRM1OPRD1OPRK1OPRL1KMT2A
SCHEMBL11133605 0.73 KDM4E (0.38) ALDH1A1OPRM1OPRD1OPRK1OPRL1
SCHEMBL9842210 0.72 OPRD1 (0.38) SLC6A9OPRM1OPRD1OPRK1KMT2A
SCHEMBL24359261 0.71 KMT2A (0.48) CNR1CNR2HTTNPSR1KMT2A
SCHEMBL5685743 0.71 ALDH1A1 (0.47) ALDH1A1CNR1CNR2HTTNPSR1
SCHEMBL5685739 0.71 ALDH1A1 (0.47) ALDH1A1CNR1CNR2HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4686217-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS FISONS PLC (GB) 1987-08-11 US disclosed
US-4607041-A CARDIOTONIC AGENTS FISONS PLC (GB) 1986-08-19 US disclosed
EP-0125803-A2 Pharmaceutically active dihydropyridines FISONS plc (GB) 1984-11-21 EP disclosed