SCHEMBL7428659

SCHEMBL7428659

OC1(CCCc2ccc(F)c(C(F)(F)F)c2)CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.42
GPR4 P46093 1/20 0.41
KCNH2 Q12809 1/20 0.41
NR3C2 P08235 1/20 0.38
AR P10275 2/20 0.38
SOS1 Q07889 1/20 0.37
PTPN7 P35236 3/20 0.36
DUSP3 P51452 3/20 0.36
SLC6A4 P31645 1/20 0.35
P2RX7 Q99572 3/20 0.35
EPHX1 P07099 1/20 0.34
GPR183 P32249 1/20 0.34
HTR1A P08908 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
HRH2 P25021 1/20 0.33
HTR1D P28221 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5498980 0.86 GPR84 (0.46) TACR1GPR4KCNH2SLC6A4P2RX7
SCHEMBL5500050 0.85 KCNH2 (0.43) TACR1GPR4KCNH2OPRM1OPRK1
Hydrochloric Acid SCHEMBL7983042 0.84 KCNH2 (0.42) TACR1GPR4KCNH2OPRM1OPRK1
SCHEMBL5502520 0.82 KCNH2 (0.41) TACR1GPR4KCNH2SOS1SLC6A4
SCHEMBL5500263 0.79 KCNH2 (0.41) TACR1GPR4KCNH2SLC6A4OPRM1
SCHEMBL5499921 0.78 IDO1 (0.43) SLC6A4P2RX7HTR1ADRD2DRD4
SCHEMBL7498985 0.78 GPR4 (0.45) TACR1GPR4KCNH2SLC6A4HTR1A
SCHEMBL5502309 0.77 KCNH2 (0.38) TACR1GPR4KCNH2SLC6A4OPRM1
Hydrochloric Acid SCHEMBL7983376 0.76 GPR4 (0.44) TACR1GPR4KCNH2SLC6A4HTR1A
SCHEMBL5495685 0.76 DPP4 (0.39) GPR4KCNH2DRD2OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1240143-A1 NEW MODULATORS OF DOPAMINE NEUROTRANSMISSION A. Carlsson Research AB (SE) 2002-09-18 EP disclosed
WO-2001046146-A1 NEW MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2001-06-28 WO disclosed