SCHEMBL7429348

SCHEMBL7429348

CC(C)C(NC(=O)OCc1ccccc1)C(O)C(F)(F)C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 7/20 0.52
CTSL P07711 6/20 0.52
CTSK P43235 8/20 0.51
ELANE P08246 2/20 0.50
ATM Q13315 1/20 0.50
CTSB P07858 4/20 0.48
PRTN3 P24158 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CTRB1 P17538 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7399913 1.00 CTSS (0.52) CTSSCTSLCTSKELANEATM
SCHEMBL5704553 0.91 CTSL (0.53) CTSSCTSLCTSKELANEATM
SCHEMBL7438056 0.90 ELANE (0.48) CTSSCTSLCTSKELANEATM
SCHEMBL10432161 0.86 CTSK (0.48) CTSSCTSLCTSKELANEATM
SCHEMBL7429948 0.85 CTSS (0.46) CTSSCTSLCTSKELANEATM
SCHEMBL12906609 0.85 ATM (0.61) CTSSCTSLCTSKELANEATM
SCHEMBL10432394 0.84 CTSK (0.46) CTSSCTSLCTSKELANEATM
SCHEMBL7296754 0.84 CTSK (0.57) CTSSCTSLCTSKCTSB
SCHEMBL10445815 0.83 CTSS (0.47) CTSSCTSLCTSKELANEATM
SCHEMBL7321385 0.82 TRPM8 (0.55) CTSSCTSLCTSKCTSBCTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114927-A Hypotensive agents and inhibiting renin MERRELL DOW PHARMACEUTICALS INC. (US) 1992-05-19 US disclosed
EP-0371179-A1 Novel analogs of peptidase substrates MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-06 EP disclosed
EP-0368719-A2 Novel analogs of peptidase substrates MERRELL PHARMACEUTICALS INC. (US) 1990-05-16 EP disclosed
EP-0362002-A1 HIV protease inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1990-04-04 EP disclosed
EP-0356595-A1 Novel peptidase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1990-03-07 EP disclosed
EP-0275101-A2 Novel peptidase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1988-07-20 EP disclosed