SCHEMBL7433951

SCHEMBL7433951

CCc1c(C)c2ccc(Oc3cccc(-c4noc(C)n4)c3)cc2[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 3/20 0.43
RAB9A P51151 2/20 0.43
HTT P42858 2/20 0.43
NPC1 O15118 1/20 0.43
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PIK3CD O00329 1/20 0.41
PIK3CB P42338 1/20 0.41
DAO P14920 1/20 0.40
HTR6 P50406 1/20 0.38
TSHR P16473 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
HPGD P15428 2/20 0.36
TUBB4A P04350 2/20 0.36
TUBB P07437 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7426351 0.82 L3MBTL1 (0.49) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7424249 0.77 LMNA (0.46) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7428004 0.77 HCRTR1 (0.44) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7428987 0.76 LMNA (0.43) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7430617 0.76 L3MBTL1 (0.49) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7538643 0.73 F2 (0.40) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7424909 0.72 L3MBTL1 (0.44) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7425441 0.71 L3MBTL1 (0.60) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7421268 0.69 MAPT (0.60) L3MBTL1LMNARAB9AHTTNPC1
SCHEMBL7430625 0.68 NQO2 (0.50) L3MBTL1LMNARAB9AHTTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107954-A1 2-OXO-$i(2H)-QUINOLINE DERIVATIVES MERCK PATENT GmbH (DE) 2001-06-20 EP disclosed
WO-2000012479-A1 2-OXO-2H-QUINOLINE DERIVATIVES MERCK PATENT GMBH (DE) 2000-03-09 WO disclosed