SCHEMBL7434190

SCHEMBL7434190

O=C(CNCc1ccccc1)Nc1cccc2[nH]ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.56
ROCK2 O75116 1/20 0.55
ROCK1 Q13464 1/20 0.55
PKN2 Q16513 1/20 0.55
DRD2 P14416 1/20 0.52
DRD4 P21917 1/20 0.52
DRD3 P35462 1/20 0.52
LMNA P02545 1/20 0.48
MAPK1 P28482 1/20 0.48
DHPS P49366 2/20 0.46
RECQL P46063 1/20 0.46
TRPV1 Q8NER1 1/20 0.45
HTT P42858 1/20 0.44
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPK14 Q16539 1/20 0.43
GSK3B P49841 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4107305 0.82 KDM4E (0.66) ALDH1A1ROCK2LMNAMAPK1DHPS
SCHEMBL29175354 0.77 LMNA (0.49) ALDH1A1LMNAHDAC3HDAC1MAPT
SCHEMBL7442891 0.77 ALDH1A1 (0.53) ALDH1A1LMNAMAPK1DHPSKDM4E
SCHEMBL25120814 0.76 DHPS (0.57) MAPK1DHPSTRPV1HDAC3HDAC1
SCHEMBL4865366 0.76 MAPK1 (0.56) ALDH1A1LMNAMAPK1DHPSTRPV1
SCHEMBL7447586 0.76 DRD4 (0.60) DRD2DRD4DRD3MAPK1GAA
SCHEMBL4025098 0.76 MAPK1 (0.63) MAPK1DHPSTRPV1
SCHEMBL29901215 0.76 MAPK1 (0.63) MAPK1DHPSTRPV1
SCHEMBL29175327 0.75 PTGS2 (0.52) ALDH1A1LMNAHDAC3HDAC1NPC1
SCHEMBL257380 0.74 MAPK1 (0.71) ALDH1A1MAPK1DHPSTRPV1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6228880-B1 PARKINSON*S DISEASE, TOURETTE*S SYNDROME, SCHIZOPHRENIA, ALCOHOLISM, DRUG ABUSE; SIDE EFFECT REDUCTION AMERICAN HOME PRODUCTS CORP 2001-05-08 US disclosed
EP-1073636-A1 4-AMINO-(ETHYLAMINO)-OXINDOLE DOPAMINE AUTORECEPTOR AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 2001-02-07 EP disclosed
WO-1999052870-A1 4-AMINO-(ETHYLAMINO)-OXINDOLE DOPAMINE AUTORECEPTOR AGONISTS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-10-21 WO disclosed