SCHEMBL7435902

SCHEMBL7435902

CN1C2CCC1CC(NC(=O)c1c(O)c3ccccc3[nH]c1=O)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.72
NPC1 O15118 3/20 0.72
MEN1 O00255 3/20 0.72
HTR3E A5X5Y0 4/20 0.70
HTR3B O95264 4/20 0.70
HTR3A P46098 4/20 0.70
HTR3D Q70Z44 4/20 0.70
HTR3C Q8WXA8 4/20 0.70
RAB9A P51151 4/20 0.68
SMN1; SMN2 Q16637 2/20 0.68
POLB P06746 2/20 0.68
RXFP1 Q9HBX9 1/20 0.68
KDM4E B2RXH2 6/20 0.57
NLRP3 Q96P20 1/20 0.57
LMNA P02545 2/20 0.54
MAPT P10636 2/20 0.54
ALDH1A1 P00352 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444121 0.97 NPC1 (0.71) KMT2ANPC1MEN1HTR3EHTR3B
SCHEMBL7300915 0.81 HTR3E (0.52) KMT2ANPC1MEN1HTR3EHTR3B
SCHEMBL22639784 0.81 RAB9A (1.00) KMT2ANPC1MEN1RAB9ASMN1; SMN2
SCHEMBL1622809 0.81 RAB9A (1.00) KMT2ANPC1MEN1RAB9ASMN1; SMN2
SCHEMBL7430312 0.81 HTR3A (0.58) KMT2AMEN1HTR3EHTR3BHTR3A
SCHEMBL7301719 0.81 HTR3E (0.51) KMT2ANPC1MEN1HTR3EHTR3B
SCHEMBL13597998 0.79 KMT2A (0.82) KMT2ANPC1MEN1RAB9ASMN1; SMN2
SCHEMBL7308018 0.78 HTR3A (0.50) KMT2ANPC1MEN1HTR3EHTR3B
SCHEMBL7430595 0.76 HTR3A (0.67) NPC1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7430349 0.75 HTR3A (1.00) NPC1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458636-B1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO KK (JP) 1995-07-12 EP disclosed
US-5248684-A CERTAIN 2-OXO-QUINOLINE CARBOXYLATES OR CORRESPONDING CARBOXAMIDES USEFUL AS ANTI-EMETICS AND SUPPRESSANTS OF MIGRAINE KYOWA HAKKO KOGYO CO., LTD. (JP) 1993-09-28 US disclosed
EP-0458636-A1 Antiemetic and migraine suppressing heterocyclic compounds and pharmaceutical compositions containing them KYOWA HAKKO KOGYO CO., LTD (JP) 1991-11-27 EP disclosed