SCHEMBL7437010

SCHEMBL7437010

CCOC(=O)C1=C(C)NC(=S)NC1c1cccc([N+](=O)[O-])c1

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.77
L3MBTL1 Q9Y468 1/20 0.74
GUSB P08236 1/20 0.74
CACNA1F O60840 9/20 0.69
CACNA1D Q01668 9/20 0.69
CACNA1S Q13698 9/20 0.69
CACNA1C Q13936 9/20 0.69
ADORA3 P0DMS8 1/20 0.69
LMNA P02545 2/20 0.69
DHFR P00374 1/20 0.68
HIF1A Q16665 3/20 0.64
MEN1 O00255 2/20 0.64
CYP1A2 P05177 2/20 0.64
CYP3A4 P08684 2/20 0.64
CYP2C9 P11712 2/20 0.64
CYP2C19 P33261 2/20 0.64
KMT2A Q03164 2/20 0.64
MAPT P10636 2/20 0.64
POLB P06746 1/20 0.64
MAPK1 P28482 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19752716 0.88 ALDH1A1 (0.71) ALDH1A1L3MBTL1CACNA1FCACNA1DCACNA1S
SCHEMBL29531249 0.88 ALDH1A1 (0.71) ALDH1A1L3MBTL1CACNA1FCACNA1DCACNA1S
SCHEMBL3394058 0.88 ALDH1A1 (0.71) ALDH1A1L3MBTL1CACNA1FCACNA1DCACNA1S
SCHEMBL7265815 0.85 ALDH1A1 (0.83) ALDH1A1L3MBTL1GUSBCACNA1FCACNA1D
Monastrol SCHEMBL3168349 0.83 KIF11 (0.77) ALDH1A1GUSBDHFRKMT2APOLB
S-Menastrol SCHEMBL74457 0.83 KIF11 (0.77) ALDH1A1GUSBDHFRKMT2APOLB
SCHEMBL14164085 0.82 DHFR (0.74) ALDH1A1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL13302798 0.82 DHFR (0.74) ALDH1A1GUSBLMNADHFRMEN1
SCHEMBL14164090 0.82 DHFR (0.74) ALDH1A1LMNADHFRKMT2APOLB
SCHEMBL2574894 0.82 CACNA1F (1.00) CACNA1FCACNA1DCACNA1SCACNA1CADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9738615-B2 Cyclophilin D inhibitors THE UNIVERSITY OF KANSAS (US) 2017-08-22 US disclosed
US-20160075669-A1 CYCLOPHILIN D INHIBITORS THE UNIVERSITY OF KANSAS 2016-03-17 US disclosed
US-4675321-A CARDIOVASCULAR DISORDERS MERCK & CO., INC. (US) 1987-06-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160075669-A1 CYCLOPHILIN D INHIBITORS PPID, APP, PIN1 ALDH1A1 2677/4885L3MBTL1 4134/4885GUSB 1712/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.