S-Menastrol

S-Menastrol

SCHEMBL74457

CCOC(=O)C1=C(C)NC(=S)N[C@H]1c1cccc(O)c1

nearest known ligand 0.77

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.77
DHFR P00374 3/20 0.76
GUSB P08236 1/20 0.70
CA1 P00915 4/20 0.64
CA2 P00918 4/20 0.64
ALDH1A1 P00352 6/20 0.63
ADORA2B P29275 4/20 0.63
POLB P06746 3/20 0.63
CA12 O43570 1/20 0.60
CA7 P43166 1/20 0.60
CA9 Q16790 1/20 0.60
KMT2A Q03164 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Monastrol SCHEMBL3168349 1.00 KIF11 (0.77) KIF11DHFRGUSBCA1CA2
SCHEMBL14164069 0.89 DHFR (0.66) KIF11DHFRGUSBCA1CA2
SCHEMBL3341613 0.87 KIF11 (0.62) KIF11DHFRGUSBCA1CA2
SCHEMBL14164085 0.87 DHFR (0.74) KIF11DHFRCA1CA2ALDH1A1
SCHEMBL13302798 0.87 DHFR (0.74) KIF11DHFRGUSBCA1CA2
SCHEMBL14164090 0.87 DHFR (0.74) KIF11DHFRCA1CA2ALDH1A1
SCHEMBL3433120 0.87 DHFR (0.64) KIF11DHFRGUSBCA1CA2
SCHEMBL5341216 0.87 KIF11 (1.00) KIF11ALDH1A1ADORA2BPOLB
SCHEMBL14164096 0.86 KIF11 (0.61) KIF11DHFRGUSBCA1CA2
SCHEMBL3343668 0.86 KIF11 (0.61) KIF11DHFRGUSBCA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 999 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024239018-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR TREATING CHEMOTHERAPY-INDUCED PERIPHERAL NEUROPATHY WITH EG5 INHIBITORS UNIVERSITY OF MIAMI (US) 2024-11-21 WO claimed
US-20240342179-A1 TREATMENT OF CANCERS OR NEOPLASMS BY INHIBITING KIF15 UNIVERSITY OF KANSAS 2024-10-17 US claimed
CN-118501443-A Preparation method of glass slide for evaluating chromosome ploidy and structure of mammal ovum 汕头市中心医院 2024-08-16 CN claimed
US-11845055-B2 Swellable organically modified silica as nanoreactors APPALACHIAN STATE UNIVERSITY (US) 2023-12-19 US claimed
US-20220008887-A1 Swellable Organically Modified Silica as Nanoreactors APPALACHIAN STATE UNIVERSITY 2022-01-13 US claimed
CN-111358792-A Application of Kif11 inhibitor monastrol in inhibiting pathological pain 中国人民解放军第四军医大学 2020-07-03 CN claimed
EP-2964625-B1 QUINOLINE SULFONYL DERIVATIVES AND USES THEREOF HEALTH SCIENCES NORTH RES INSTITUTE (CA) 2018-07-25 EP claimed
US-9975852-B2 Quinoline sulfonyl derivatives and uses thereof HEALTH SCIENCES NORTH RESEARCH INSTITUTE (CA) 2018-05-22 US claimed
US-20160298168-A1 PROTEIN STRUCTURAL BIOMARKERS TO GUIDE TARGETED CHEMOTHERAPIES KIM SUNYOUNG (US) 2016-10-13 US claimed
EP-2399136-B1 PROTEIN STRUCTURAL BIOMARKERS TO GUIDE TARGETED CHEMOTHERAPIES KIM SUNYOUNG (US) 2016-06-22 EP claimed
WO-2010096680-A2 PROTEIN STRUCTURAL BIOMARKERS TO GUIDE TARGETED CHEMOTHERAPIES BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL COLLEGE (US) 2010-08-26 WO claimed
CN-101781259-A Precursor compound of 18F marked tumor inhibitor Monastrol as well as preparation method and application UNIV ZHEJIANG 2010-07-21 CN claimed
EP-2188630-A2 METHODS AND COMPOSITIONS RELATED TO SYNERGISTIC RESPONSES TO ONCOGENIC MUTATIONS THE UNIVERSITY OF ROCHESTER (US) 2010-05-26 EP claimed
EP-2182986-A2 ANTI-MITOTIC AGENT AND AURORA KINASE INHIBITOR COMBINATION AS ANTI-CANCER TREATMENT SCHERING CORPORATION (US) 2010-05-12 EP claimed
US-20100016252-A1 Mannich Base N-Oxide Drugs State of Oregon Acting By and Through The Oregon State Board of Higher Education On Behalf of The U (US) 2010-01-21 US claimed
EP-2136626-A1 MANNICH BASE N-OXIDE DRUGS State of Oregon acting by and through the Oregon State Board of Higher Education on behalf of the University of Oregon (US) 2009-12-30 EP claimed
WO-2009099991-A2 TREATMENT OF CANCER THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2009-08-13 WO claimed
WO-2009045443-A2 METHODS AND COMPOSITIONS RELATED TO SYNERGISTIC RESPONSES TO ONCOGENIC MUTATIONS THE UNIVERSITY OF ROCHESTER (US) 2009-04-09 WO claimed
WO-2009017701-A2 ANTI-MITOTIC AGENT AND AURORA KINASE INHIBITOR COMBINATION AS ANTI-CANCER TREATMENT SCHERING CORPORATION (US) 2009-02-05 WO claimed
WO-2008115499-A1 MANNICH BASE N-OXIDE DRUGS STATE OF OREGON ACTING BY AND THROUGH THE OREGON STATE BOARD OF HIGHER EDUCATION ON BEHALF OF THE UNIVERSITY OF OREGON (US) 2008-09-25 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11845055-B2 Swellable organically modified silica as nanoreactors MSN, SORD, OGA KIF11 1028/4885DHFR 1319/4885GUSB 349/4885
US-20220008887-A1 Swellable Organically Modified Silica as Nanoreactors MSN, SORD, OGA KIF11 1028/4885DHFR 1319/4885GUSB 349/4885
US-20100016252-A1 Mannich Base N-Oxide Drugs ASAH2, MAN2B1, NNT KIF11 2056/4885DHFR 540/4885GUSB 229/4885
US-20240342179-A1 TREATMENT OF CANCERS OR NEOPLASMS BY INHIBITING KIF15 KIF15, KIF11, KIF2C KIF11 2/4885DHFR 993/4885GUSB 4191/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.