SCHEMBL7437290

SCHEMBL7437290

COC(=O)CN1Cc2ccc([N+](=O)[O-])cc2CNC1=O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PNMT P11086 7/20 0.42
ADRA2A P08913 5/20 0.42
ADRA2B P18089 2/20 0.42
ADRA2C P18825 2/20 0.42
DPP7 Q9UHL4 1/20 0.41
NAMPT P43490 1/20 0.41
ALDH1A1 P00352 2/20 0.40
GLA P06280 1/20 0.40
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434141 0.95 ITGB3 (0.41) PNMTADRA2AADRA2BADRA2CDPP7
SCHEMBL7440791 0.76 ITGB3 (0.47) NAMPTALDH1A1
SCHEMBL7664159 0.76 ALDH1A1 (0.42) DPP7NAMPTALDH1A1GLANPC1
SCHEMBL7448788 0.74 ALDH1A1 (0.42) DPP7NAMPTALDH1A1GLANPC1
SCHEMBL655730 0.74 ALDH1A1 (0.44) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL655452 0.74 ALDH1A1 (0.41) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL14558962 0.73 DRD2 (0.54) ALDH1A1NPC1MAPTMAPK1RAB9A
SCHEMBL7399767 0.71 ALDH1A1 (0.40) PNMTADRA2AADRA2BADRA2CALDH1A1
SCHEMBL38658114 0.71 DPP7 (0.51) DPP7NAMPTALDH1A1GLAMAPT
SCHEMBL8699228 0.70 SIRT2 (0.48) ALDH1A1NPC1MAPTMAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403578-B1 ANTICOAGULANTS, CARDIOVASCULAR DISORDERS SMITHKLINE BEECHAM CORPORATION 2002-06-11 US disclosed
EP-0674623-A1 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1995-10-04 EP disclosed
WO-1994014776-A2 BICYCLIC FIBRINOGEN ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1994-07-07 WO disclosed