SCHEMBL7438142

SCHEMBL7438142

Clc1ccccc1N1[CH]CNCC1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.59
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
HTR1A P08908 5/20 0.40
HTR3A P46098 4/20 0.40
CYP1A2 P05177 3/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C9 P11712 3/20 0.40
ALOX5 P09917 2/20 0.40
RXFP1 Q9HBX9 1/20 0.39
SLC6A2 P23975 1/20 0.38
HTR7 P34969 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
PLA2G1B P04054 1/20 0.37
RAB9A P51151 1/20 0.37
ATG4B Q9Y4P1 1/20 0.37
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6352703 0.86 DRD2 (0.60) ADRB1DRD2DRD3HTR1AHTR3A
SCHEMBL2414713 0.79 HTR1A (0.39) ADRB1HTR1AHTR3ASLC6A2HTR7
SCHEMBL2209185 0.79 ADRB1 (0.58) ADRB1DRD2DRD3HTR1AHTR3A
SCHEMBL5785574 0.75 ADRB1 (1.00) ADRB1DRD2DRD3HTR1AHTR3A
SCHEMBL29446047 0.75 ADRB1 (1.00) ADRB1DRD2DRD3HTR1AHTR3A
SCHEMBL230424 0.75 ADRB1 (1.00) ADRB1DRD2DRD3HTR1AHTR3A
SCHEMBL3483188 0.75 DRD2 (0.61) ADRB1DRD2DRD3HTR1AHTR3A
SCHEMBL8357275 0.75 EPHX2 (0.44) ADRB1HTR1AHTR3ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL29777392 0.73 ADRB1 (0.96) ADRB1DRD2DRD3HTR1AHTR3A
Hydrochloric Acid SCHEMBL6577765 0.73 ADRB1 (0.96) ADRB1DRD2DRD3HTR1AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454501-B1 Benzylidenethiazolidine derivatives, their preparation and their use for the inhibition of lipid peroxides SANKYO CO (JP) 2001-09-05 EP disclosed
EP-0839812-A1 Preparation of benzylthiazolidine derivatives Sankyo Company Limited (JP) 1998-05-06 EP disclosed
EP-0479665-A2 1,4-Dihydropyridine derivatives, method for preparing the same and use thereof TEIKOKU CHEMICAL INDUSTRIES CO., LTD. (JP) 1992-04-08 EP disclosed
EP-0454501-A2 Benzylidenethiazolidine derivatives, their preparation and their use for the inhibition of lipid peroxides Sankyo Company Limited (JP) 1991-10-30 EP disclosed