SCHEMBL7444030

SCHEMBL7444030

O=C(O)CC1C(=O)NCc2cc(C(=O)O)ccc2N1CCc1ccc2c(c1)OCO2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.43
ALDH1A1 P00352 6/20 0.40
MAPK1 P28482 1/20 0.40
ITGB3 P05106 2/20 0.39
ITGAV P06756 2/20 0.39
SRD5A2 P31213 1/20 0.38
PTGER4 P35408 1/20 0.38
PTGER2 P43116 1/20 0.38
TSHR P16473 3/20 0.37
NAAA Q02083 1/20 0.36
PDE5A O76074 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
KDM4E B2RXH2 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TAS2R14 Q9NYV8 1/20 0.35
SSTR5 P35346 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078805 0.75 TSHR (0.43) ALDH1A1ITGB3ITGAVTSHRKDM4E
SCHEMBL7366389 0.75 TSHR (0.43) ALDH1A1ITGB3ITGAVTSHRKDM4E
SCHEMBL7079518 0.75 TSHR (0.36) ALDH1A1ITGB3TSHRKDM4ETDP1
SCHEMBL7397950 0.74 ALDH1A1 (0.52) ALDH1A1TSHRKDM4ESMN1; SMN2
SCHEMBL7132139 0.71 ITGB3 (0.67) ITGB3ITGAV
SCHEMBL7333012 0.71 TSHR (0.39) ALDH1A1ITGB3ITGAVTSHRKDM4E
SCHEMBL27720182 0.67 ALDH1A1 (0.67) HPGDALDH1A1MAPK1SRD5A2PTGER4
Piperonylic Acid SCHEMBL3936749 0.65 ALDH1A1 (0.73) HPGDALDH1A1MAPK1SRD5A2PDE5A
Piperonylic Acid SCHEMBL142318 0.63 ALDH1A1 (1.00) HPGDALDH1A1MAPK1SRD5A2MEN1
Piperonylic Acid SCHEMBL31119409 0.63 ALDH1A1 (1.00) HPGDALDH1A1MAPK1SRD5A2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0767792-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-11-20 EP disclosed
EP-0767792-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-04-16 EP disclosed
WO-1996000730-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-01-11 WO disclosed