SCHEMBL7444159

SCHEMBL7444159

CCc1ccccc1S(=O)(=O)NCc1cc(O)c(C(c2cccc(NS(=O)(=O)c3cccc4cccnc34)c2)C2CC2)c(=O)o1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.42
ALDH1A1 P00352 5/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
PKM P14618 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
TRPV1 Q8NER1 1/20 0.39
BRD4 O60885 1/20 0.39
HPGD P15428 1/20 0.39
FABP1 P07148 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
GHSR Q92847 1/20 0.39
ADRA1A P35348 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432825 0.87 NAMPT (0.38) KMT2AGAABRD4
SCHEMBL7441054 0.87 ALOX12 (0.37) PDE4BALDH1A1GAAHTT
SCHEMBL7448162 0.84 HSP90AA1 (0.39) ALDH1A1LMNAMEN1KMT2ATDP1
SCHEMBL7450441 0.84 ALOX12 (0.39) ALDH1A1LMNAMEN1KMT2A
SCHEMBL7444165 0.84 PDE4B (0.40) PDE4BALDH1A1LMNAMEN1KMT2A
SCHEMBL7437309 0.83 ALOX12 (0.36) ALDH1A1LMNATDP1MAPTHTT
SCHEMBL7445966 0.83 TACR1 (0.34) ALDH1A1KMT2APKMMAPT
SCHEMBL7437636 0.82 ATIC (0.36) BRD4
SCHEMBL6174502 0.82 PDE4B (0.42) PDE4BALDH1A1LMNAMEN1KMT2A
SCHEMBL7445646 0.82 ALDH1A1 (0.35) ALDH1A1LMNAMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed