SCHEMBL7450441

SCHEMBL7450441

CCc1ccccc1S(=O)(=O)NCc1cc(O)c(C(c2cccc(NS(=O)(=O)c3ccc(F)cc3)c2)C2CC2)c(=O)o1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 6/20 0.39
HSP90AA1 P07900 2/20 0.36
HSP90AB1 P08238 2/20 0.36
HSD17B3 P37058 1/20 0.35
HSD17B2 P37059 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
ATM Q13315 1/20 0.34
KMT2A Q03164 3/20 0.33
LMNA P02545 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PGAM1 P18669 1/20 0.33
MEN1 O00255 2/20 0.33
MAPK14 Q16539 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441054 0.94 ALOX12 (0.37) ALOX12ALDH1A1
SCHEMBL7437309 0.91 ALOX12 (0.36) ALOX12LMNAPGAM1ALDH1A1
SCHEMBL7437636 0.91 ATIC (0.36) ALOX12HSD17B2PGAM1
Ethane SCHEMBL7484090 0.90 ALOX12 (0.38) ALOX12HSP90AA1HSP90AB1HSD17B3HSD17B2
SCHEMBL7432825 0.88 NAMPT (0.38) ALOX12HSD17B2KMT2A
SCHEMBL7448162 0.85 HSP90AA1 (0.39) HSP90AA1HSP90AB1L3MBTL1KMT2ALMNA
Ethane SCHEMBL7480930 0.85 POLB (0.39) ALOX12KMT2AMEN1ALDH1A1
SCHEMBL7445966 0.85 TACR1 (0.34) KMT2AALDH1A1
SCHEMBL7444159 0.84 PDE4B (0.42) KMT2ALMNAMEN1ALDH1A1
SCHEMBL7445646 0.84 ALDH1A1 (0.35) KMT2ALMNAMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed