SCHEMBL7445966

SCHEMBL7445966

CCc1ccccc1S(=O)(=O)NCc1cc(O)c(C(c2ccccc2)C2CC2)c(=O)o1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.34
KMT2A Q03164 1/20 0.34
PKM P14618 1/20 0.33
CTSB P07858 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 2/20 0.32
MCL1 Q07820 2/20 0.32
CYP2C9 P11712 1/20 0.32
BCL2L1 Q07817 1/20 0.32
MAPT P10636 1/20 0.31
ACHE P22303 1/20 0.31
KCNK3 O14649 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441054 0.89 ALOX12 (0.37) ALDH1A1POLB
SCHEMBL7445646 0.85 ALDH1A1 (0.35) KMT2AALDH1A1POLBMAPT
SCHEMBL7450441 0.85 ALOX12 (0.39) KMT2AALDH1A1
SCHEMBL7437309 0.84 ALOX12 (0.36) ALDH1A1MCL1MAPT
SCHEMBL7432825 0.84 NAMPT (0.38) KMT2A
SCHEMBL7448162 0.84 HSP90AA1 (0.39) KMT2AALDH1A1POLBMAPT
SCHEMBL7437636 0.83 ATIC (0.36)
SCHEMBL7444159 0.83 PDE4B (0.42) KMT2APKMALDH1A1MAPT
SCHEMBL6177695 0.78 CYP2C9 (0.38) KMT2AALDH1A1CYP2C9MAPT
Ethane SCHEMBL7480930 0.78 POLB (0.39) KMT2AALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed