SCHEMBL7448162

SCHEMBL7448162

CCc1ccccc1S(=O)(=O)NCc1cc(O)c(C(c2cccc(NS(=O)(=O)c3cc(Cl)ccc3Cl)c2)C2CC2)c(=O)o1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 6/20 0.39
HSP90AB1 P08238 6/20 0.39
MAPT P10636 4/20 0.36
TP53 P04637 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HSD11B1 P28845 1/20 0.35
DPP4 P27487 1/20 0.35
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ITGA1 P56199 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethane SCHEMBL7485196 0.90 HSP90AA1 (0.39) HSP90AA1HSP90AB1MAPTTP53ALDH1A1
SCHEMBL7441054 0.88 ALOX12 (0.37) ALDH1A1HTTPOLB
SCHEMBL7450441 0.85 ALOX12 (0.39) HSP90AA1HSP90AB1ALDH1A1LMNAL3MBTL1
SCHEMBL7444159 0.84 PDE4B (0.42) MAPTALDH1A1LMNAHTTTDP1
SCHEMBL7432825 0.84 NAMPT (0.38) KMT2A
SCHEMBL7437309 0.84 ALOX12 (0.36) MAPTALDH1A1LMNAHTTTDP1
SCHEMBL7445966 0.84 TACR1 (0.34) MAPTALDH1A1POLBKMT2A
SCHEMBL7437636 0.84 ATIC (0.36) HSD11B1
SCHEMBL7445646 0.83 ALDH1A1 (0.35) MAPTALDH1A1LMNATDP1HSD17B10
SCHEMBL7448164 0.82 ALDH1A1 (0.40) HSP90AA1HSP90AB1MAPTTP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed