SCHEMBL7444252

SCHEMBL7444252

CCOC(=O)[C@@]1(c2ccc(OC)cc2)COS(=O)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
HTT P42858 2/20 0.40
KMT2A Q03164 4/20 0.39
MEN1 O00255 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 3/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
HPGD P15428 4/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 1/20 0.38
GLA P06280 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439116 1.00 ALDH1A1 (0.40) ALDH1A1HTTKMT2AMEN1L3MBTL1
SCHEMBL7442579 0.87 L3MBTL1 (0.37) ALDH1A1KMT2AMEN1L3MBTL1POLB
SCHEMBL7442583 0.87 L3MBTL1 (0.37) ALDH1A1KMT2AMEN1L3MBTL1POLB
SCHEMBL14967672 0.84 ALDH1A1 (0.43) ALDH1A1HTTKMT2AMEN1L3MBTL1
SCHEMBL21874111 0.77 ALDH1A1 (0.39) ALDH1A1HTTKMT2AMEN1L3MBTL1
SCHEMBL21874235 0.74 LMNA (0.46) ALDH1A1KMT2AMEN1L3MBTL1POLB
SCHEMBL14968165 0.73 CHRM1 (0.44) ALDH1A1KMT2AMEN1POLBCYP2C9
SCHEMBL14967816 0.72 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1L3MBTL1POLB
SCHEMBL28318807 0.72 OPRM1 (0.57) LMNASMN1; SMN2NPSR1TDP1CHRM2
SCHEMBL5166279 0.70 OPRM1 (0.51) KMT2AMEN1CYP2C9CYP2C19LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5869697-A Process for preparing diltiazem COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 1999-02-09 US claimed
US-6180785-B1 REFLUXING AMINOTHIOPHENOL OR AMINOTHIONAPHTHOL WITH ALKOXYPHENYL-4-CARBOALKOXY-1,3,2-DIOXATHIOLANE COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2001-01-30 US disclosed
US-5869697-A Process for preparing diltiazem COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 1999-02-09 US disclosed