SCHEMBL7444401

SCHEMBL7444401

Nc1c(NCc2ccccc2)ccn(CC(=O)N2CCCCC2)c1=O

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 3/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 3/20 0.42
PREP P48147 1/20 0.42
NPC1 O15118 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
PTGS2 P35354 1/20 0.41
PPID Q08752 1/20 0.40
GRIN2B Q13224 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9179794 0.78 GRM2 (0.43) KDM4ESMN1; SMN2MAPTNPC1GRIN2B
Hydrochloric Acid SCHEMBL8993826 0.71 ALDH1A1 (0.51) ALDH1A1KDM4ETSHRSMN1; SMN2KMT2A
SCHEMBL9478463 0.69 MAPT (0.41) POLBMAPT
SCHEMBL9184025 0.68 CASP3 (0.44) ALDH1A1KDM4ESMN1; SMN2POLB
SCHEMBL7444409 0.67 KMT2A (0.41) ALDH1A1KDM4ESMN1; SMN2POLBKMT2A
SCHEMBL29518393 0.67 LTA4H (0.57) ALDH1A1POLBKMT2ANPC1TDP1
SCHEMBL27829698 0.66 KMT2A (0.60) ALDH1A1KDM4ESMN1; SMN2POLBKMT2A
SCHEMBL14597067 0.66 KCNQ2 (0.50) ALDH1A1TSHRKMT2AMAPT
SCHEMBL10381350 0.65 LTA4H (0.58) ALDH1A1KDM4EPOLBKMT2ANPC1
SCHEMBL18050010 0.64 LOXL2 (0.57) ALDH1A1KDM4ETSHRSMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5438063-A Hypotensive agents, cardiac insufficiency, increased intraocular pressure, and CNS disorders MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-08-01 US disclosed
EP-0628556-A1 Imidazopyridines MERCK PATENT GmbH (DE) 1994-12-14 EP disclosed