SCHEMBL7451104

SCHEMBL7451104

CCCC[SiH2]OC(c1ccccc1)(c1ccccc1)c1cc(C=O)cc(C(=O)O)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UNG P13051 1/20 0.36
PLA2G2A P14555 1/20 0.33
STS P08842 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31
NPC1 O15118 1/20 0.31
CYP2C9 P11712 1/20 0.31
RAB9A P51151 1/20 0.31
ALDH1A1 P00352 2/20 0.31
S1PR3 Q99500 1/20 0.31
TSHR P16473 2/20 0.30
TRIM24 O15164 1/20 0.30
TRIM33 Q9UPN9 1/20 0.30
TP53 P04637 1/20 0.30
HDAC3 O15379 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC2 Q92769 1/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
CA2 P00918 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447426 0.83 PRKCA (0.36) PLA2G2A
SCHEMBL6170855 0.80 UNG (0.40) UNGALDH1A1TRIM24TRIM33TP53
SCHEMBL7510342 0.78 MEN1 (0.41) NPC1CYP2C9RAB9AALDH1A1TSHR
SCHEMBL10544293 0.66 SMN1; SMN2 (0.50) UNGNPC1RAB9AALDH1A1TRIM24
SCHEMBL2997840 0.66 CES2 (0.48) UNGNPC1RAB9AALDH1A1TRIM24
SCHEMBL2773374 0.65 PLA2G2A (0.65) PLA2G2ATSHRTP53
SCHEMBL12813482 0.64 KIF11 (0.50) CYP2C9
SCHEMBL6172247 0.64 PRKCA (0.38) NPC1RAB9ATSHRTP53HSD17B10
SCHEMBL6170678 0.62 TSHR (0.41) NPSR1RAB9AALDH1A1TSHRKDM4E
SCHEMBL3470017 0.62 UNG (0.61) UNGALDH1A1TSHRTRIM24TRIM33

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192127-A1 SUBSTITUTED BENZAMIDE INHIBITORS OF RHINOVIRUS 3C PROTEASE Agouron Pharmaceuticals, Inc. (US) 2002-04-03 EP disclosed
WO-2000078708-A1 SUBSTITUTED BENZAMIDE INHIBITORS OF RHINOVIRUS 3C PROTEASE AGOURON PHARMACEUTICALS, INC. (US) 2000-12-28 WO disclosed