SCHEMBL7453262

SCHEMBL7453262

O=[C]C(CNC=O)c1cccs1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
KEAP1 Q14145 1/20 0.33
MAPT P10636 1/20 0.32
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31
ADH1B P00325 2/20 0.31
ADH1C P00326 2/20 0.31
ADH1A P07327 2/20 0.31
ADH7 P40394 1/20 0.31
ALOX5 P09917 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453266 0.77 LMNA (0.36) LMNACES2CES1KEAP1MAPT
SCHEMBL7456996 0.75 CTSC (0.38) CES2CES1KEAP1MAPTTP53
SCHEMBL144586 0.74 ALOX5 (0.38) LMNACES2CES1KEAP1MAPT
SCHEMBL142885 0.71 TAS1R3 (0.36) LMNACES2CES1KEAP1MAPT
SCHEMBL11314837 0.70 FFAR1 (0.46) LMNACES2CES1KEAP1MAPT
SCHEMBL141982 0.69 HTT (0.40) LMNACES2CES1KEAP1MAPT
SCHEMBL11169009 0.68 HTT (0.36) LMNACES2CES1KEAP1MAPT
SCHEMBL10458682 0.67 ALOX5 (0.43) LMNACES2CES1KEAP1MAPT
SCHEMBL11309726 0.66 CES2 (0.36) CES2CES1KEAP1MAPTALOX5
SCHEMBL7534282 0.66 SMN1; SMN2 (0.38) LMNATP53POLBADH1BADH1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001027096-A9 AMINOMETHYL-(HETERO)ARYL DERIVATIVES AND THEIR USE AS TRYPTASE INHIBITORS PROTHERICS MOLECULAR DESIGN LT (GB) 2001-07-12 WO disclosed