SCHEMBL7464951

SCHEMBL7464951

Cc1c[nH]c(-c2nc(C(=O)CC(=O)Nc3cc(-c4ccccc4F)ccc3NC(=O)O)cs2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.41
LMNA P02545 1/20 0.40
MAOA P21397 1/20 0.38
HDAC1 Q13547 3/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC3 O15379 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
LDHA P00338 1/20 0.34
GHSR Q92847 1/20 0.34
DHODH Q02127 2/20 0.34
RAB9A P51151 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
EIF4E P06730 1/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464517 0.90 ACHE (0.36) ACHELMNAMAOAHDAC1HDAC8
SCHEMBL7459709 0.78 KCNQ4 (0.37) LMNAHDAC1HDAC8HDAC3HDAC6
SCHEMBL7466556 0.71 ADCY8 (0.38) HDAC1HDAC8HDAC3HDAC7HDAC6
SCHEMBL5869160 0.70 LDHA (0.37) HDAC1HDAC3HDAC6LDHAMAPT
SCHEMBL7465533 0.70 KAT6A (0.37) LMNAMAOAHDAC1HDAC8HDAC3
SCHEMBL7531659 0.66 MAPT (0.56) LMNAMEN1MAPTKMT2AALDH1A1
SCHEMBL7707033 0.65 HPGDS (0.38) ACHEMAOAHDAC1HDAC3HDAC6
SCHEMBL5563091 0.63 CYP17A1 (0.41)
SCHEMBL5559220 0.63 CYP17A1 (0.39) HDAC1HDAC3HDAC6RAB9ASMN1; SMN2
SCHEMBL2693403 0.62 ACHE (0.63) ACHELMNAHDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224175-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029012-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed