SCHEMBL7464956

SCHEMBL7464956

COc1ccc2cc(C(=O)Nc3ccc4[nH]c(C(=O)N5C[C@@H](CCl)c6c5cc(O)c5[nH]c(C(F)(F)F)c(C(=O)O)c65)cc4c3)oc2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.35
NPC1 O15118 5/20 0.35
RAB9A P51151 5/20 0.35
ALDH1A1 P00352 2/20 0.35
PRNP P04156 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MAPT P10636 5/20 0.34
KMT2A Q03164 3/20 0.34
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
MEN1 O00255 2/20 0.32
TP53 P04637 2/20 0.32
TSHR P16473 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
APP P05067 1/20 0.32
ACHE P22303 1/20 0.32
AKR1C3 P42330 1/20 0.31
CYP2D6 P10635 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7465517 0.95 KDM4E (0.36) KDM4ENPC1RAB9AALDH1A1PRNP
SCHEMBL7471301 0.90 CNR1 (0.31) KDM4ENPC1MAPTKMT2AMEN1
SCHEMBL7468511 0.89 HRH4 (0.36) KDM4ENPC1RAB9AALDH1A1PRNP
SCHEMBL7475427 0.89 KMT2A (0.33) KDM4ENPC1RAB9AMAPTKMT2A
SCHEMBL6627433 0.89 MAPT (0.38) KDM4ENPC1RAB9AMAPTKMT2A
SCHEMBL7460763 0.88 KDM4E (0.37) KDM4ENPC1RAB9AALDH1A1PRNP
SCHEMBL7467710 0.88 KMT2A (0.36) KDM4ENPC1RAB9AALDH1A1L3MBTL1
SCHEMBL7473569 0.88 P4HB (0.34) KDM4EMAPT
SCHEMBL7463553 0.87 KDM4E (0.36) KDM4ENPC1RAB9AALDH1A1PRNP
SCHEMBL7474728 0.87 MGLL (0.35) NPC1RAB9AAPPACHECYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656360-B1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-11-20 EP disclosed
US-5629430-A ANTICARCINOGENIC AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-05-13 US disclosed
EP-0656360-A1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1995-06-07 EP disclosed