SCHEMBL7474728

SCHEMBL7474728

COc1ccc2cc(C(=O)N3C[C@@H](CCl)c4c3cc(O)c3[nH]c(C(F)(F)F)c(C(=O)O)c43)oc2c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.35
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 2/20 0.33
SLC16A3 O15427 1/20 0.32
APP P05067 2/20 0.32
ACHE P22303 1/20 0.32
RAB9A P51151 2/20 0.32
HRH3 Q9Y5N1 3/20 0.31
ADH1A P07327 1/20 0.31
KIT P10721 1/20 0.31
FLT1 P17948 1/20 0.31
FLT4 P35916 1/20 0.31
KDR P35968 1/20 0.31
ABL2 P42684 1/20 0.31
NPC1 O15118 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470246 0.94 HRH3 (0.34) HRH3
SCHEMBL7464956 0.87 KDM4E (0.35) CYP2D6APPACHERAB9ANPC1
SCHEMBL7470331 0.86 LMNA (0.36) RAB9ANPC1
SCHEMBL7463040 0.85 ADH1A (0.33) ACHEADH1AKITFLT1FLT4
SCHEMBL7474788 0.84 P4HB (0.34)
SCHEMBL7465517 0.82 KDM4E (0.36) APPACHERAB9ANPC1
SCHEMBL7465748 0.79 ALDH1A1 (0.37) CYP1A2CYP2D6ACHERAB9ANPC1
SCHEMBL7465921 0.79 ALDH1A1 (0.37) CYP1A2CYP2D6ACHERAB9ANPC1
SCHEMBL13401627 0.79 TAS1R3 (0.37)
SCHEMBL7465950 0.78 AKR1C3 (0.39) RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656360-B1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-11-20 EP disclosed
US-5629430-A ANTICARCINOGENIC AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-05-13 US disclosed
EP-0656360-A1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1995-06-07 EP disclosed