Beclomethasone Dipropionate

Beclomethasone Dipropionate

SCHEMBL74651

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nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Beclomethasone Dipropionate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 6/20 0.94
CYP3A4 P08684 8/20 0.94
USP2 O75604 6/20 0.94
PGR P06401 5/20 0.94
HIF1A Q16665 4/20 0.94
ADORA3 P0DMS8 3/20 0.94
AR P10275 2/20 0.94
CNR1 P21554 2/20 0.94
CHRM1 P11229 1/20 0.94
TBXA2R P21731 1/20 0.94
MAPT P10636 3/20 0.76
NR1I2 O75469 2/20 0.76
DRD2 P14416 1/20 0.76
OPRD1 P41143 1/20 0.76
LMNA P02545 5/20 0.65
ABCB11 O95342 4/20 0.65
CYP2C9 P11712 3/20 0.65
CYP2D6 P10635 2/20 0.65
SMN1; SMN2 Q16637 2/20 0.65
MLNR O43193 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Beclomethasone Dipropionate SCHEMBL14782876 0.99 CYP3A4 (0.95) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL7329 0.99 CYP3A4 (0.95) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL1216647 0.98 CYP3A4 (0.98) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL74650 0.98 CYP3A4 (0.98) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL3930413 0.97 CYP3A4 (0.91) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL6890 0.97 CYP3A4 (1.00) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL10392062 0.97 CYP3A4 (1.00) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL2404673 0.97 CYP3A4 (1.00) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL9768491 0.97 CYP3A4 (1.00) CYP3A4USP2NR3C1PGRHIF1A
Beclomethasone Dipropionate SCHEMBL13653326 0.97 CYP3A4 (1.00) CYP3A4USP2NR3C1PGRHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 972 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210401798-A1 LIPOXIN A4 ANALOGS AND USES THEREOF THE BRIGHAM AND WOMEN'S HOSPITAL, INC. (US) 2021-12-30 US claimed
CN-113795246-A Injectable sustained release formulation for the treatment of joint pain and inflammation 福多兹制药公司 2021-12-14 CN claimed
US-20210177866-A1 PROCESS FOR PREPARING A DRY POWDER FORMULATION COMPRISING AN ANTICHOLINERGIC, A CORTICOSTEROID AND A BETA-ADRENERGIC CHIESI FARMACEUTICI S.P.A. (IT) 2021-06-17 US claimed
US-10966991-B2 Process for preparing a dry powder formulation comprising an anticholinergic, a corticosteroid and a beta-adrenergic CHIESI FARMACEUTICI S.P.A. (IT) 2021-04-06 US claimed
US-20200368252-A1 PROCESS FOR PREPARING A DRY POWDER FORMULATION COMPRISING AN ANTICHOLINERGIC, A CORTICOSTEROID AND A BETA-ADRENERGIC CHIESI FARMMACEUTICI S.P.A. (IT) 2020-11-26 US claimed
US-10772896-B2 Process for preparing a dry powder formulation comprising an anticholinergic, a corticosteroid and a beta-adrenergic CHIESI FARMACEUTICI S.P.A. (IT) 2020-09-15 US claimed
US-10548864-B2 Enhanced ATRA-related compounds for the treatment of proliferative diseases, autoimmune diseases, and addiction conditions BETH ISRAEL DEACONESS MEDICAL CENTER, INC. (US) 2020-02-04 US claimed
US-20180360849-A1 PROCESS FOR PREPARING A DRY POWDER FORMULATION COMPRISING AN ANTICHOLINERGIC, A CORTICOSTEROID AND A BETA-ADRENERGIC CHIESI FARMACEUTICI S.P.A. (IT) 2018-12-20 US claimed
US-10086004-B2 Process for preparing a dry powder formulation comprising an anticholinergic, a corticosteroid and a beta-adrenergic CHIESI FARMACEUTICI S.P.A. (IT) 2018-10-02 US claimed
US-20180064666-A1 ENHANCED ATRA-RELATED COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES, AUTOIMMUNE DISEASES, AND ADDICTION CONDITIONS BETH ISRAEL DEACONESS MEDICAL CENTER, INC. 2018-03-08 US claimed
EP-1073417-A1 PHARMACEUTICAL AEROSOL FORMULATION GLAXO GROUP LIMITED (GB) 2001-02-07 EP claimed
US-6149892-A INHALER HAVING INTERIOR SURFACES COATED WITH BLEND OF FLUOROPOLYMER(S) AND NON-FLUOROPOLYMER(S) AND CONTAINING ACTIVE DRUG AND A FLUOROCARBON PROPELLANT; ACCURATE DRUG DELIVERY GLAXOWELLCOME, INC. (US) 2000-11-21 US claimed
CN-1048394-C Medicaments GLAXO GROUP LTD (GB) 2000-01-19 CN claimed
WO-1999053901-A1 PHARMACEUTICAL AEROSOL FORMULATION GLAXO GROUP LIMITED (GB) 1999-10-28 WO claimed
CN-1186473-A Metered dose inhaler for beclomethasone dipropionate GLAXO WELLCOME INC (US) 1998-07-01 CN claimed
US-5695744-A Medicaments GLAXO GROUP LIMITED (GB) 1997-12-09 US claimed
US-5688782-A Medicaments for treating respiratory disorders GLAXO GROUP LIMITED (GB) 1997-11-18 US claimed
EP-0625046-B1 Pharmaceutical aerosol formulations comprising beclomethasone dipropionate GLAXO GROUP LTD (GB) 1997-09-10 EP claimed
CN-1078633-A pharmaceutical preparation GLAXO GROUP LTD (GB) 1993-11-24 CN claimed
US-4866051-A TREATMENT OR PROPHYLAXIS OF ASTHMA; INHALANTS GLAXO GROUP LIMITED (GB) 1989-09-12 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210401798-A1 LIPOXIN A4 ANALOGS AND USES THEREOF LTA4H, ALOX15B, LTB4R NR3C1 736/4885CYP3A4 423/4885USP2 4225/4885
US-10548864-B2 Enhanced ATRA-related compounds for the treatment of proliferative diseases, autoimmune diseases, and addiction conditions PIN1, RARB, RARA NR3C1 290/4885CYP3A4 3907/4885USP2 2626/4885
US-20180064666-A1 ENHANCED ATRA-RELATED COMPOUNDS FOR THE TREATMENT OF PROLIFERATIVE DISEASES, AUTOIMMUNE DISEASES, AND ADDICTION CONDITIONS PIN1, RARB, RARA NR3C1 290/4885CYP3A4 3907/4885USP2 2626/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.