SCHEMBL7466337

SCHEMBL7466337

CC(=O)NOC(=O)CCNC(=O)c1cccc(N2CCC(Nc3ncccn3)CC2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.43
CNR2 P34972 1/20 0.43
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 1/20 0.41
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
KDR P35968 2/20 0.38
DRD4 P21917 3/20 0.38
PDGFRB P09619 1/20 0.38
DRD2 P14416 3/20 0.38
DRD3 P35462 3/20 0.38
VCP P55072 2/20 0.38
PLOD2 O00469 1/20 0.37
PLOD3 O60568 1/20 0.37
PLOD1 Q02809 1/20 0.37
F10 P00742 1/20 0.37
HSD17B10 Q99714 1/20 0.37
EPHX2 P34913 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6496334 0.90 CNR1 (0.43) CNR1CNR2HDAC3HDAC1KDM4E
SCHEMBL6503936 0.89 CNR1 (0.41) CNR1CNR2HDAC3HDAC1KDM4E
SCHEMBL7464413 0.89 CNR1 (0.45) CNR1CNR2HDAC3HDAC1KDM4E
SCHEMBL7467073 0.86 VCP (0.41) CNR1CNR2HDAC3HDAC1KDM4E
SCHEMBL7457979 0.84 SFRP1 (0.42) CNR1CNR2KDM4EHTTDRD4
SCHEMBL7468782 0.82 DRD4 (0.42) CNR1CNR2HTTDRD4DRD2
SCHEMBL381765 0.81 ALDH1A1 (0.46) CNR1CNR2HDAC1KDM4EHTT
SCHEMBL6499244 0.79 CNR1 (0.38) CNR1CNR2HDAC3HDAC1KDM4E
SCHEMBL382963 0.79 SMYD3 (0.43) CNR1CNR2HDAC3HDAC1KDM4E
SCHEMBL6499974 0.78 ITGB3 (0.43) CNR1CNR2HDAC1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1229024-A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRIN ALPHA-V BETA-3 ANTAGONISM MEIJI SEIKA KAISHA LTD. (JP) 2002-08-07 EP claimed
EP-1229024-A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRIN ALPHA-V BETA-3 ANTAGONISM MEIJI SEIKA KAISHA LTD. (JP) 2002-08-07 EP disclosed