SCHEMBL7467178

SCHEMBL7467178

N#CC(=Cc1cc2ccccc2cn1)C(=O)Nc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.56
MEN1 O00255 5/20 0.56
KDM4E B2RXH2 4/20 0.56
ALDH1A1 P00352 8/20 0.54
MAPT P10636 8/20 0.54
MAPK1 P28482 4/20 0.54
LMNA P02545 4/20 0.54
HPGD P15428 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
CYP1A2 P05177 2/20 0.54
CYP2C19 P33261 2/20 0.54
PKM P14618 2/20 0.54
TDP1 Q9NUW8 2/20 0.54
PSMD14 O00487 1/20 0.54
RGS12 O14924 1/20 0.54
GMNN O75496 1/20 0.54
EGFR P00533 1/20 0.54
ERBB2 P04626 1/20 0.54
TP53 P04637 1/20 0.54
CYP3A4 P08684 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7461493 0.92 MAPT (0.48) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7470135 0.82 LMNA (0.62) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7463147 0.80 MCL1 (0.53) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7463154 0.80 MCL1 (0.53) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7461370 0.80 ALDH1A1 (0.59) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7470342 0.77 MEN1 (0.60) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7463673 0.75 ALDH1A1 (0.53) KMT2AMEN1KDM4EALDH1A1MAPT
Tyrphostin Ag 494 SCHEMBL15362064 0.75 KMT2A (0.74) KMT2AMEN1KDM4EALDH1A1MAPT
Tyrphostin Ag 494 SCHEMBL20645572 0.75 KMT2A (0.74) KMT2AMEN1KDM4EALDH1A1MAPT
SCHEMBL7181057 0.73 RAB9A (0.73) KMT2AMEN1KDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700388-B1 SUBSTITUTED BETA-ARYL AND BETA-HETEROARYL-ALPHA-CYANOACRYLAMIDE DERIVATIVES AS TYROSINE KINASE INHIBITORS PHARMACIA ITALIA SPA (IT) 2002-09-18 EP claimed