SCHEMBL7470321

SCHEMBL7470321

N=C(N)NCCc1ccc(OCCC2Oc3cc([N+](=O)[O-])ccc3N(Cc3ccccc3Cl)C2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPFFR1 Q9GZQ6 1/20 0.36
NPFFR2 Q9Y5X5 1/20 0.36
ALDH1A1 P00352 8/20 0.36
MAPT P10636 3/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
KCNH2 Q12809 1/20 0.35
MEN1 O00255 5/20 0.34
KMT2A Q03164 5/20 0.34
TP53 P04637 2/20 0.34
CYP1A2 P05177 1/20 0.34
ALOX15 P16050 1/20 0.34
MAPK1 P28482 1/20 0.34
RECQL P46063 1/20 0.34
CACNA1C Q13936 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PKM P14618 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7462740 0.99 NPFFR1 (0.36) NPFFR1NPFFR2ALDH1A1MAPTTSHR
SCHEMBL8605543 0.96 NPFFR1 (0.36) NPFFR1NPFFR2ALDH1A1MAPTTSHR
SCHEMBL8554026 0.91 KCNH2 (0.41) ALDH1A1MAPTKCNH2MEN1KMT2A
SCHEMBL7476790 0.90 TSHR (0.45) ALDH1A1TSHRHTTTP53
SCHEMBL8551402 0.89 MEN1 (0.39) ALDH1A1MAPTTSHRKCNH2MEN1
SCHEMBL8604248 0.88 ALDH1A1 (0.38) ALDH1A1MAPTTSHRHTTKCNH2
SCHEMBL8556736 0.88 SIRT2 (0.41) ALDH1A1MAPTTSHRKCNH2MEN1
Hydrochloric Acid SCHEMBL8602861 0.88 MEN1 (0.39) ALDH1A1MAPTKCNH2MEN1KMT2A
SCHEMBL7466586 0.88 PTPN1 (0.38) ALDH1A1MAPTTSHRKCNH2MEN1
SCHEMBL8555600 0.85 SIRT2 (0.43) ALDH1A1MAPTTSHRHTTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869949-B1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO MCNEIL PHARM INC (US) 2002-12-18 EP claimed
EP-0869949-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1998-10-14 EP disclosed
WO-1997017333-A1 BENZOXAZINE ANTIMICROBIAL AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1997-05-15 WO disclosed