SCHEMBL7474018

SCHEMBL7474018

COc1ccc(CCc2ccc(F)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.60
MEN1 O00255 1/20 0.60
POLB P06746 1/20 0.60
MAPT P10636 1/20 0.60
MAPK1 P28482 1/20 0.60
KMT2A Q03164 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
TAAR1 Q96RJ0 1/20 0.59
ALDH1A1 P00352 1/20 0.58
NFE2L2 Q16236 1/20 0.57
FPR2 P25090 1/20 0.55
TUBB4A P04350 1/20 0.55
TUBB P07437 1/20 0.55
TUBA3C P0DPH7 1/20 0.55
TUBA1B P68363 1/20 0.55
TUBA4A P68366 1/20 0.55
TUBB4B P68371 1/20 0.55
TUBB3 Q13509 1/20 0.55
TUBB2A Q13885 1/20 0.55
TUBB8 Q3ZCM7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL834551 0.88 TAAR1 (0.73) TAAR1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3794098 0.86 LTA4H (0.65) KDM4EMEN1POLBMAPTMAPK1
SCHEMBL8298 0.85
SCHEMBL7024215 0.85
SCHEMBL9973127 0.85 ALDH1A1 (0.61) KDM4EMEN1POLBMAPTMAPK1
SCHEMBL10450398 0.81 TAAR1 (0.64) TAAR1TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL20767237 0.81 LMNA (0.67) KDM4EMEN1POLBMAPTMAPK1
SCHEMBL21340442 0.81 MAOB (0.69) POLBMAOB
SCHEMBL1304164 0.80 NPC1 (0.71) KDM4EMEN1MAPTKMT2AL3MBTL1
SCHEMBL4435722 0.80 MAPT (0.62) KDM4EMEN1POLBMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110437230-A A kind of three-level aminated compounds and biphosphine ligand, wherein mesosome and preparation method SHANGHAI INST ORGANIC CHEMISTRY CAS 2019-11-12 CN disclosed
WO-2007045366-A1 HETEROCYCLIC COMPOUNDS WITH CARBOXYL ISOSTERE GROUPS AND THEIR USE FOR THE TREATMENT OF CARDIOVASCULAR DISEASES BAYER HEALTHCARE AG (DE) 2007-04-26 WO disclosed
EP-1206474-A1 SULFONYLPHENYLPYRAZOLE COMPOUNDS USEFUL AS COX-2 INHIBITORS ABBOTT LABORATORIES (US) 2002-05-22 EP disclosed
WO-2001016138-A1 SULFONYLPHENYLPYRAZOLE COMPOUNDS USEFUL AS COX-2 INHIBITORS ABBOTT LABORATORIES (US) 2001-03-08 WO disclosed