SCHEMBL7475931

SCHEMBL7475931

CCOC(=O)[C@H](Cc1ccc2c(c1)NC(=O)[C@@H](CCCNC(=O)OCc1ccccc1)O2)NS(=O)(=O)c1c(C)c(C)cc(C)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.42
HSD17B10 Q99714 3/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
MMP2 P08253 3/20 0.38
MMP9 P14780 3/20 0.38
BACE1 P56817 1/20 0.38
USP2 O75604 2/20 0.36
TSHR P16473 2/20 0.35
MAPT P10636 1/20 0.35
MMP1 P03956 1/20 0.35
MMP3 P08254 1/20 0.35
MMP7 P09237 1/20 0.35
MMP13 P45452 1/20 0.35
AVPR1B P47901 1/20 0.35
ACE P12821 1/20 0.35
THRB P10828 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7163466 0.95 MMP2 (0.42) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7374585 0.92 MMP2 (0.44) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7364535 0.89 ALOX15 (0.41) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7479990 0.88 HSD17B10 (0.40) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7365624 0.87 CASP1 (0.41) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7364118 0.87 ALOX15 (0.43) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7474783 0.85 ITGB3 (0.44) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7164959 0.85 MMP2 (0.51) IDO1TDO2MMP2MMP9MMP1
SCHEMBL7479315 0.84 ALOX15 (0.41) ALOX15HSD17B10MAPK1HTTL3MBTL1
SCHEMBL7478564 0.83 ALOX15 (0.44) ALOX15HSD17B10MAPK1HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964856-B1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 2002-10-09 EP disclosed