SCHEMBL7364535

SCHEMBL7364535

CCOC(=O)[C@H](Cc1ccc2c(c1)NC(=O)[C@@H](CCCNC(=O)OCc1ccccc1)O2)NS(=O)(=O)Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 3/20 0.41
HSD17B10 Q99714 3/20 0.41
L3MBTL1 Q9Y468 3/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
IDO1 P14902 2/20 0.40
TDO2 P48775 1/20 0.40
ITGB3 P05106 3/20 0.38
ITGAV P06756 1/20 0.38
TMPRSS11D O60235 1/20 0.38
ACE P12821 1/20 0.38
ITGA2B P08514 2/20 0.37
MAPT P10636 2/20 0.37
BACE1 P56817 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7163731 0.93 ITGB3 (0.43) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7479990 0.93 HSD17B10 (0.40) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7374585 0.91 MMP2 (0.44) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7364118 0.90 ALOX15 (0.43) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7475931 0.89 ALOX15 (0.42) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7167879 0.88 ITGB3 (0.42) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7365624 0.87 CASP1 (0.41) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7479315 0.86 ALOX15 (0.41) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7478564 0.86 ALOX15 (0.44) ALOX15HSD17B10L3MBTL1MAPK1HTT
SCHEMBL7469657 0.86 MAPT (0.44) ALOX15HSD17B10L3MBTL1MAPK1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0964856-B1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 2002-10-09 EP disclosed
EP-0964856-A1 BICYCLIC AMINO ACIDS MERCK PATENT GmbH (DE) 1999-12-22 EP disclosed
WO-1998035949-A1 BICYCLIC AMINO ACIDS MERCK PATENT GMBH (DE) 1998-08-20 WO disclosed